Insights into the cellular pharmacological properties of the BET-inhibitor OTX015/MK-8628 (birabresib), alone and in combination, in leukemia models.

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Title: Insights into the cellular pharmacological properties of the BET-inhibitor OTX015/MK-8628 (birabresib), alone and in combination, in leukemia models.
Authors: Astorgues-Xerri, Lucile1 (AUTHOR), Vázquez, Ramiro2 (AUTHOR), Odore, Elodie3 (AUTHOR), Rezai, Keyvan3 (AUTHOR), Kahatt, Carmen1 (AUTHOR), Mackenzie, Sarah1 (AUTHOR), Bekradda, Mohamed1 (AUTHOR), Coudé, Marie-Magdelaine4 (AUTHOR), Dombret, Herve4 (AUTHOR), Gardin, Claude4 (AUTHOR), Lokiec, Francois3 (AUTHOR), Raymond, Eric5 (AUTHOR), Noel, Kay6 (AUTHOR), Cvitkovic, Esteban6 (AUTHOR), Herait, Patrice6 (AUTHOR), Bertoni, Francesco2 (AUTHOR) frbertoni@mac.com, Riveiro, María E.1 (AUTHOR) eugenia.riveiro@e2dg.com
Source: Leukemia & Lymphoma. Dec2019, Vol. 60 Issue 12, p3067-3070. 4p.
Database: Academic Search Ultimate
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ISSN:10428194
DOI:10.1080/10428194.2019.1617860