The antischistosomal potential of GSK-J4, an H3K27 demethylase inhibitor: insights from molecular modeling, transcriptomics and in vitro assays.

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Title: The antischistosomal potential of GSK-J4, an H3K27 demethylase inhibitor: insights from molecular modeling, transcriptomics and in vitro assays.
Authors: Lobo-Silva, Jessica1 (AUTHOR), Cabral, Fernanda J.2 (AUTHOR), Amaral, Murilo S.3 (AUTHOR), Miyasato, Patrícia A.4 (AUTHOR), de Freitas, Rafaela Paula4 (AUTHOR), Pereira, Adriana S. A.3,5 (AUTHOR), Khouri, Mariana I.1 (AUTHOR), Barbosa, Mayra M. F.6 (AUTHOR), Ramos, Pablo I. P.7 (AUTHOR), Leite, Luciana C. C.6 (AUTHOR), Asojo, Oluwatoyin A.8 (AUTHOR), Nakano, Eliana4 (AUTHOR), Verjovski-Almeida, Sergio3,5 (AUTHOR), Farias, Leonardo P.1 (AUTHOR) leonardo.farias@bahia.fiocruz.br
Source: Parasites & Vectors. 3/17/2020, Vol. 13 Issue 1, p1-16. 16p.
Database: Academic Search Ultimate
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ISSN:17563305
DOI:10.1186/s13071-020-4000-z