DNA-Dependent Protein Kinase (DNA-PK) Inhibitors. Synthesis and Biological Activity of Quinolin-4-one and Pyridopyrimidin-4-one Surrogates for the Chromen-4-one Chemotype.

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Title: DNA-Dependent Protein Kinase (DNA-PK) Inhibitors. Synthesis and Biological Activity of Quinolin-4-one and Pyridopyrimidin-4-one Surrogates for the Chromen-4-one Chemotype.
Authors: Cano, Céline1,2 (AUTHOR) celine.cano@ncl.ac.uk, Barbeau, Olivier R.2 (AUTHOR), Bailey, Christine3 (AUTHOR), Cockcroft, Xiao-Ling3 (AUTHOR), Curtin, Nicola J.2 (AUTHOR), Duggan, Heather3 (AUTHOR), Frigerio, Mark3 (AUTHOR), Golding, Bernard T.2 (AUTHOR), Hardcastle, Ian R.2 (AUTHOR), Hummersone, Marc G.3 (AUTHOR), Knights, Charlotte3 (AUTHOR), Menear, Keith A.3 (AUTHOR), Newell, David R.2 (AUTHOR), Richardson, Caroline J.3 (AUTHOR), Smith, Graeme C. M.3 (AUTHOR), Spittle, Ben3 (AUTHOR), Griffin, Roger J.2 (AUTHOR)
Source: Journal of Medicinal Chemistry. 12/23/2010, Vol. 53 Issue 24, p8498-8507. 10p.
Database: Academic Search Ultimate
Description
ISSN:00222623
DOI:10.1021/jm100608j