An FDA-Approved Antifungal, Ketoconazole, and Its Novel Derivative Suppress tGLI1-Mediated Breast Cancer Brain Metastasis by Inhibiting the DNA-Binding Activity of Brain Metastasis-Promoting Transcription Factor tGLI1.

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Title: An FDA-Approved Antifungal, Ketoconazole, and Its Novel Derivative Suppress tGLI1-Mediated Breast Cancer Brain Metastasis by Inhibiting the DNA-Binding Activity of Brain Metastasis-Promoting Transcription Factor tGLI1.
Authors: Doheny, Daniel1 (AUTHOR), Manore, Sara1 (AUTHOR), Sirkisoon, Sherona R.1 (AUTHOR), Zhu, Dongqin1 (AUTHOR), Aguayo, Noah R.1 (AUTHOR), Harrison, Alexandria1 (AUTHOR), Najjar, Mariana1 (AUTHOR), Anguelov, Marlyn1 (AUTHOR), Cox, Anderson O'Brien2 (AUTHOR), Furdui, Cristina M.2,3,4 (AUTHOR), Watabe, Kounosuke1,4 (AUTHOR), Hollis, Thomas4,5 (AUTHOR), Thomas, Alexandra4,6 (AUTHOR), Strowd, Roy4,7 (AUTHOR), Lo, Hui-Wen1,4 (AUTHOR) hlo@wakehealth.edu
Source: Cancers. Sep2022, Vol. 14 Issue 17, p4256. 21p.
Database: Academic Search Ultimate
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ISSN:20726694
DOI:10.3390/cancers14174256