Towards Translation of PqsR Inverse Agonists: From In Vitro Efficacy Optimization to In Vivo Proof‐of‐Principle.

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Title: Towards Translation of PqsR Inverse Agonists: From In Vitro Efficacy Optimization to In Vivo Proof‐of‐Principle.
Authors: Hamed, Mostafa M.1,2 (AUTHOR), Abdelsamie, Ahmed S.1,2,3 (AUTHOR), Rox, Katharina2,4 (AUTHOR), Schütz, Christian1,2 (AUTHOR), Kany, Andreas M.1,2 (AUTHOR), Röhrig, Teresa1,2 (AUTHOR), Schmelz, Stefan5 (AUTHOR), Blankenfeldt, Wulf5,6 (AUTHOR), Arce‐Rodriguez, Alejandro7 (AUTHOR), Borrero‐de Acuña, José Manuel7,8,9 (AUTHOR), Jahn, Dieter7,8 (AUTHOR), Rademacher, Jessica10,11 (AUTHOR), Ringshausen, Felix C.10,11,12 (AUTHOR), Cramer, Nina13 (AUTHOR), Tümmler, Burkhard11,13 (AUTHOR), Hirsch, Anna K. H.1,2,14 (AUTHOR), Hartmann, Rolf W.1,2,14 (AUTHOR), Empting, Martin1,2,14 (AUTHOR) Martin.empting@helmholtz-hzi.de
Source: Advanced Science. 2/14/2023, Vol. 10 Issue 5, p1-14. 14p.
Database: Academic Search Ultimate
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ISSN:21983844
DOI:10.1002/advs.202204443