Discovery of arylsulfonamides as a novel class of allosteric integrase inhibitors with antiviral activity.
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| Title: | Discovery of arylsulfonamides as a novel class of allosteric integrase inhibitors with antiviral activity. |
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| Authors: | Wang, Cheng1 (AUTHOR), Adam, Gregory C.2 (AUTHOR), Burlein, Christine3 (AUTHOR), Carroll, Steven3 (AUTHOR), Dankulich, William1 (AUTHOR), Diamond, Tracy4 (AUTHOR), Grobler, Jay4 (AUTHOR), Heath, Jeffrey4 (AUTHOR), Johnson, Adam1 (AUTHOR), Klein, Daniel5 (AUTHOR), Krosky, Daniel3 (AUTHOR), Narayan, Kartik3 (AUTHOR), Ou, Yangsi3 (AUTHOR), Sanders, John5 (AUTHOR), Sharma, Sujata2 (AUTHOR), Xu, Min3 (AUTHOR), Converso, Antonella1 (AUTHOR) antonella_converso@merck.com |
| Source: | Bioorganic & Medicinal Chemistry Letters. Jun2023, Vol. 89, pN.PAG-N.PAG. 1p. |
| Database: | Academic Search Ultimate |
| ISSN: | 0960894X |
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| DOI: | 10.1016/j.bmcl.2023.129303 |