Discovery of the First‐in‐Class Inhibitors of Hypoxia Up‐Regulated Protein 1 (HYOU1) Suppressing Pathogenic Fibroblast Activation.

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Title: Discovery of the First‐in‐Class Inhibitors of Hypoxia Up‐Regulated Protein 1 (HYOU1) Suppressing Pathogenic Fibroblast Activation.
Authors: Papadopoulou, Dimitra1 (AUTHOR), Mavrikaki, Vasiliki2,3 (AUTHOR), Charalampous, Filippos1 (AUTHOR), Tzaferis, Christos1 (AUTHOR), Samiotaki, Martina1 (AUTHOR), Papavasileiou, Konstantinos D.4,5,6 (AUTHOR), Afantitis, Antreas4,5,6 (AUTHOR), Karagianni, Niki7 (AUTHOR), Denis, Maria C.7 (AUTHOR), Sanchez, Julie8,9 (AUTHOR), Lane, J. Robert8,9 (AUTHOR), Faidon Brotzakis, Zacharias1,10 (AUTHOR), Skretas, Georgios1,11 (AUTHOR), Georgiadis, Dimitris3 (AUTHOR), Matralis, Alexios N.1 (AUTHOR) matralis@fleming.gr, Kollias, George1,12,13 (AUTHOR) kollias@fleming.gr
Source: Angewandte Chemie International Edition. 4/2/2024, Vol. 63 Issue 14, p1-13. 13p.
Database: Academic Search Ultimate
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ISSN:14337851
DOI:10.1002/anie.202319157