Asciminib, a novel allosteric inhibitor of BCR‐ABL1, shows synergistic effects when used in combination with imatinib with or without drug resistance.

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Title: Asciminib, a novel allosteric inhibitor of BCR‐ABL1, shows synergistic effects when used in combination with imatinib with or without drug resistance.
Authors: Okamoto, Naoki1,2, Yagi, Kenta1,3 yagi.kenta@tokushima-u.ac.jp, Imawaka, Sayaka1, Takaoka, Mayu1, Aizawa, Fuka1,2, Niimura, Takahiro1,3, Goda, Mitsuhiro1,2, Miyata, Koji1, Kawada, Kei1,4, Izawa‐Ishizawa, Yuki1,5, Sakaguchi, Satoshi3,6, Ishizawa, Keisuke1,2,3
Source: Pharmacology Research & Perspectives. Aug2024, Vol. 12 Issue 4, p1-9. 9p.
Database: Academic Search Ultimate
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ISSN:20521707
DOI:10.1002/prp2.1214