Discovery and evaluation of novel Benzohydroxamic acid-indole derivatives as dual inhibitors of ADAM17 and HDAC2 with antitumor activity.
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| Title: | Discovery and evaluation of novel Benzohydroxamic acid-indole derivatives as dual inhibitors of ADAM17 and HDAC2 with antitumor activity. |
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| Authors: | Song, Xiaoxuan1,2 (AUTHOR), Tong, Xin1 (AUTHOR), Yang, Kaisi1 (AUTHOR), Qi, Yiming1 (AUTHOR), Liu, Wenwu3 (AUTHOR), Sun, Yuzhu4 (AUTHOR), Wang, Chengkang1 (AUTHOR), Xun, Fanghua1 (AUTHOR), Wang, Ziyi1 (AUTHOR), Jiang, Muxuan1 (AUTHOR), Zhang, Yingshi5 (AUTHOR), Ren, Tianshu1 (AUTHOR), Chen, Di6,7 (AUTHOR), Hou, Shanbo8 (AUTHOR), Song, Aigang8 (AUTHOR), Gao, Huiyuan1,2,9,10 (AUTHOR) sypugaohy@163.com, Zhao, Qingchun1,2,5 (AUTHOR) zhaoqingchun1967@163.com |
| Source: | Bioorganic Chemistry. Apr2025, Vol. 157, pN.PAG-N.PAG. 1p. |
| Database: | Academic Search Ultimate |
| ISSN: | 00452068 |
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| DOI: | 10.1016/j.bioorg.2025.108308 |