Matrix Approach Assessment of Cabotegravir Drug–Drug Interactions with OAT1/OAT3 Substrates and UGT1A1/UGT1A9 Inhibitors Using Physiologically-Based Pharmacokinetic Modeling.

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Title: Matrix Approach Assessment of Cabotegravir Drug–Drug Interactions with OAT1/OAT3 Substrates and UGT1A1/UGT1A9 Inhibitors Using Physiologically-Based Pharmacokinetic Modeling.
Authors: Tracey, Helen1 (AUTHOR), Bate, Simon T.1,2 (AUTHOR), Ford, Susan2,3 (AUTHOR), Patel, Parul1,3 (AUTHOR), Bloomer, Jackie1,2 (AUTHOR), Patel, Aarti1,3 (AUTHOR), Taskar, Kunal S.1 (AUTHOR) kunal.s.taskar@gsk.com
Source: Pharmaceutics. Apr2025, Vol. 17 Issue 4, p531. 20p.
Database: Academic Search Ultimate
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ISSN:19994923
DOI:10.3390/pharmaceutics17040531