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Discovery of TNG-6132, a potent, selective, and orally bioavailable USP1 inhibitor.

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Title: Discovery of TNG-6132, a potent, selective, and orally bioavailable USP1 inhibitor.
Authors: Throner, Scott1 (AUTHOR), Feng, Tianshu1 (AUTHOR), Andersen, Jannik N.1 (AUTHOR), Bandi, Madhavi1 (AUTHOR), Engel, Justin L.1 (AUTHOR), Gong, Shanzhong1 (AUTHOR), Gotur, Deepali1 (AUTHOR), Gu, Lina1 (AUTHOR), Huang, Alan1 (AUTHOR), Lazarides, Katherine1 (AUTHOR), Maxwell, John P.1 (AUTHOR), McCarren, Patrick1 (AUTHOR), McMillan, Brian J.1 (AUTHOR), Pham, Truc V.1 (AUTHOR), Simoneau, Antoine1 (AUTHOR), Tsai, Alice1 (AUTHOR), Whittington, Douglas A.1 (AUTHOR), Wilker, Erik1 (AUTHOR), Zhang, Minjie1 (AUTHOR), Zhang, Wenhai1 (AUTHOR)
Source: Bioorganic & Medicinal Chemistry Letters. Aug2025, Vol. 124, pN.PAG-N.PAG. 1p.
Database: Academic Search Ultimate
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Header DbId: asn
DbLabel: Academic Search Ultimate
An: 185200490
AccessLevel: 2
PubType: Academic Journal
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  Data: <searchLink fieldCode="JN" term="%22Bioorganic+%26+Medicinal+Chemistry+Letters%22">Bioorganic & Medicinal Chemistry Letters</searchLink>. Aug2025, Vol. 124, pN.PAG-N.PAG. 1p.
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=185200490
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