Discovery of TNG-6132, a potent, selective, and orally bioavailable USP1 inhibitor.
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| Title: | Discovery of TNG-6132, a potent, selective, and orally bioavailable USP1 inhibitor. |
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| Authors: | Throner, Scott1 (AUTHOR), Feng, Tianshu1 (AUTHOR), Andersen, Jannik N.1 (AUTHOR), Bandi, Madhavi1 (AUTHOR), Engel, Justin L.1 (AUTHOR), Gong, Shanzhong1 (AUTHOR), Gotur, Deepali1 (AUTHOR), Gu, Lina1 (AUTHOR), Huang, Alan1 (AUTHOR), Lazarides, Katherine1 (AUTHOR), Maxwell, John P.1 (AUTHOR), McCarren, Patrick1 (AUTHOR), McMillan, Brian J.1 (AUTHOR), Pham, Truc V.1 (AUTHOR), Simoneau, Antoine1 (AUTHOR), Tsai, Alice1 (AUTHOR), Whittington, Douglas A.1 (AUTHOR), Wilker, Erik1 (AUTHOR), Zhang, Minjie1 (AUTHOR), Zhang, Wenhai1 (AUTHOR) |
| Source: | Bioorganic & Medicinal Chemistry Letters. Aug2025, Vol. 124, pN.PAG-N.PAG. 1p. |
| Database: | Academic Search Ultimate |
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