3D-QSAR Design of New Bcr-Abl Inhibitors Based on Purine Scaffold and Cytotoxicity Studies on CML Cell Lines Sensitive and Resistant to Imatinib.

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Title: 3D-QSAR Design of New Bcr-Abl Inhibitors Based on Purine Scaffold and Cytotoxicity Studies on CML Cell Lines Sensitive and Resistant to Imatinib.
Authors: Cabezas, David1 (AUTHOR), Delgado, Thalía2 (AUTHOR), Sepúlveda, Guisselle2,3 (AUTHOR), Krňávková, Petra3,4 (AUTHOR), Vojáčková, Veronika3,5 (AUTHOR), Kryštof, Vladimír3,6 (AUTHOR), Strnad, Miroslav4,7 (AUTHOR), Silva, Nicolás Ignacio2,8 (AUTHOR), Echeverría, Javier1,5 (AUTHOR), Espinosa-Bustos, Christian2,6 (AUTHOR), Mellado, Guido3,7 (AUTHOR), Luo, Jiao1,4 (AUTHOR), Mella, Jaime1,5,8 (AUTHOR), Salas, Cristian O.2,6 (AUTHOR)
Source: Pharmaceuticals (14248247). Jun2025, Vol. 18 Issue 6, p925. 27p.
Database: Academic Search Ultimate
Description
ISSN:14248247
DOI:10.3390/ph18060925