The ATM Kinase Inhibitor AZD0156 Is a Potent Inhibitor of Plasmodium Phosphatidylinositol 4‐Kinase (PI4Kβ) and Is an Attractive Candidate for Medicinal Chemistry Optimization Against Malaria.

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Title: The ATM Kinase Inhibitor AZD0156 Is a Potent Inhibitor of Plasmodium Phosphatidylinositol 4‐Kinase (PI4Kβ) and Is an Attractive Candidate for Medicinal Chemistry Optimization Against Malaria.
Authors: Woodland, John G.1,2,3 (AUTHOR), Coertzen, Dina4 (AUTHOR), Wicht, Kathryn J.1,2,3 (AUTHOR), Hidalgo, Virginia Franco5 (AUTHOR), Pasaje, Charisse Flerida A.6 (AUTHOR), Godoy, Luiz C.6 (AUTHOR), Qahash, Tarrick7,8 (AUTHOR), Mmonwa, Mmakwena M.1 (AUTHOR), Dziwornu, Godwin A.1 (AUTHOR), Wambua, Lynn2,3 (AUTHOR), Harries, Sarah3 (AUTHOR), Korkor, Constance M.3 (AUTHOR), Njoroge, Mathew1 (AUTHOR), Krugmann, Liezl1 (AUTHOR), Taylor, Dale1 (AUTHOR), Leshabane, Meta4 (AUTHOR), Langeveld, Henrico4 (AUTHOR), Rabie, Tayla4 (AUTHOR), Reader, Janette4 (AUTHOR), van der Watt, Mariëtte4 (AUTHOR)
Source: Angewandte Chemie International Edition. 7/7/2025, Vol. 64 Issue 28, p1-10. 10p.
Database: Academic Search Ultimate
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ISSN:14337851
DOI:10.1002/anie.202425206