Fragment‐Based Drug Discovery of Novel High‐affinity, Selective, and Anti‐inflammatory Inhibitors of the Keap1‐Nrf2 Protein‐Protein Interaction.

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Bibliographic Details
Title: Fragment‐Based Drug Discovery of Novel High‐affinity, Selective, and Anti‐inflammatory Inhibitors of the Keap1‐Nrf2 Protein‐Protein Interaction.
Authors: Lin, Chunyu1 (AUTHOR), Narayanan, Dilip1 (AUTHOR), Barreca, Marilia1,2 (AUTHOR), Poulsen, Cecilie3 (AUTHOR), da Costa, Leandro Silva3 (AUTHOR), Chen, Xiangrong4 (AUTHOR), Wichman, Kendall G.5 (AUTHOR), Charley, Cherisse A.5 (AUTHOR), Lindsay, Jaslin L.5 (AUTHOR), Dezfouli, Mahya6 (AUTHOR), Vlissari, Dimitra1 (AUTHOR), Mortensen, Thomas S.1 (AUTHOR), Chan, Camilla B.1,7 (AUTHOR), Wang, Jingyi1 (AUTHOR), Richardson, William4 (AUTHOR), Manning, Charlotte E.4 (AUTHOR), Chen, Zhuoyao4 (AUTHOR), Zang, Jie1 (AUTHOR), Käck, Helena8 (AUTHOR), Gajhede, Michael1 (AUTHOR)
Source: Angewandte Chemie International Edition. 9/22/2025, Vol. 64 Issue 39, p1-12. 12p.
Database: Academic Search Ultimate
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Description
ISSN:14337851
DOI:10.1002/anie.202508121