Fragment‐Based Drug Discovery of Novel High‐affinity, Selective, and Anti‐inflammatory Inhibitors of the Keap1‐Nrf2 Protein‐Protein Interaction.
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| Title: | Fragment‐Based Drug Discovery of Novel High‐affinity, Selective, and Anti‐inflammatory Inhibitors of the Keap1‐Nrf2 Protein‐Protein Interaction. |
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| Authors: | Lin, Chunyu1 (AUTHOR), Narayanan, Dilip1 (AUTHOR), Barreca, Marilia1,2 (AUTHOR), Poulsen, Cecilie3 (AUTHOR), da Costa, Leandro Silva3 (AUTHOR), Chen, Xiangrong4 (AUTHOR), Wichman, Kendall G.5 (AUTHOR), Charley, Cherisse A.5 (AUTHOR), Lindsay, Jaslin L.5 (AUTHOR), Dezfouli, Mahya6 (AUTHOR), Vlissari, Dimitra1 (AUTHOR), Mortensen, Thomas S.1 (AUTHOR), Chan, Camilla B.1,7 (AUTHOR), Wang, Jingyi1 (AUTHOR), Richardson, William4 (AUTHOR), Manning, Charlotte E.4 (AUTHOR), Chen, Zhuoyao4 (AUTHOR), Zang, Jie1 (AUTHOR), Käck, Helena8 (AUTHOR), Gajhede, Michael1 (AUTHOR) |
| Source: | Angewandte Chemie International Edition. 9/22/2025, Vol. 64 Issue 39, p1-12. 12p. |
| Database: | Academic Search Ultimate |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 188158491 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=188158491 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1002/anie.202508121 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 12 StartPage: 1 Titles: – TitleFull: Fragment‐Based Drug Discovery of Novel High‐affinity, Selective, and Anti‐inflammatory Inhibitors of the Keap1‐Nrf2 Protein‐Protein Interaction. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Lin, Chunyu – PersonEntity: Name: NameFull: Narayanan, Dilip – PersonEntity: Name: NameFull: Barreca, Marilia – PersonEntity: Name: NameFull: Poulsen, Cecilie – PersonEntity: Name: NameFull: da Costa, Leandro Silva – PersonEntity: Name: NameFull: Chen, Xiangrong – PersonEntity: Name: NameFull: Wichman, Kendall G. – PersonEntity: Name: NameFull: Charley, Cherisse A. – PersonEntity: Name: NameFull: Lindsay, Jaslin L. – PersonEntity: Name: NameFull: Dezfouli, Mahya – PersonEntity: Name: NameFull: Vlissari, Dimitra – PersonEntity: Name: NameFull: Mortensen, Thomas S. – PersonEntity: Name: NameFull: Chan, Camilla B. – PersonEntity: Name: NameFull: Wang, Jingyi – PersonEntity: Name: NameFull: Richardson, William – PersonEntity: Name: NameFull: Manning, Charlotte E. – PersonEntity: Name: NameFull: Chen, Zhuoyao – PersonEntity: Name: NameFull: Zang, Jie – PersonEntity: Name: NameFull: Käck, Helena – PersonEntity: Name: NameFull: Gajhede, Michael IsPartOfRelationships: – BibEntity: Dates: – D: 22 M: 09 Text: 9/22/2025 Type: published Y: 2025 Identifiers: – Type: issn-print Value: 14337851 Numbering: – Type: volume Value: 64 – Type: issue Value: 39 Titles: – TitleFull: Angewandte Chemie International Edition Type: main |
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