Fragment‐Based Drug Discovery of Novel High‐affinity, Selective, and Anti‐inflammatory Inhibitors of the Keap1‐Nrf2 Protein‐Protein Interaction.

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Title: Fragment‐Based Drug Discovery of Novel High‐affinity, Selective, and Anti‐inflammatory Inhibitors of the Keap1‐Nrf2 Protein‐Protein Interaction.
Authors: Lin, Chunyu1 (AUTHOR), Narayanan, Dilip1 (AUTHOR), Barreca, Marilia1,2 (AUTHOR), Poulsen, Cecilie3 (AUTHOR), da Costa, Leandro Silva3 (AUTHOR), Chen, Xiangrong4 (AUTHOR), Wichman, Kendall G.5 (AUTHOR), Charley, Cherisse A.5 (AUTHOR), Lindsay, Jaslin L.5 (AUTHOR), Dezfouli, Mahya6 (AUTHOR), Vlissari, Dimitra1 (AUTHOR), Mortensen, Thomas S.1 (AUTHOR), Chan, Camilla B.1,7 (AUTHOR), Wang, Jingyi1 (AUTHOR), Richardson, William4 (AUTHOR), Manning, Charlotte E.4 (AUTHOR), Chen, Zhuoyao4 (AUTHOR), Zang, Jie1 (AUTHOR), Käck, Helena8 (AUTHOR), Gajhede, Michael1 (AUTHOR)
Source: Angewandte Chemie International Edition. 9/22/2025, Vol. 64 Issue 39, p1-12. 12p.
Database: Academic Search Ultimate
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