Discovery of benzyl carbamate inhibitors of coronavirus Mpro enzymes from a legacy collection of cysteine protease inhibitors.

Saved in:
Bibliographic Details
Title: Discovery of benzyl carbamate inhibitors of coronavirus Mpro enzymes from a legacy collection of cysteine protease inhibitors.
Authors: Sá Magalhães Serafim, Mateus1,2,3 (AUTHOR), Kronenberger, Thales4,5 (AUTHOR), Francisco, Karol R.1 (AUTHOR), de Sousa Reis, Erik Vinicius2 (AUTHOR), Gonçalves de Oliveira, Ellen1,2 (AUTHOR), Marcelino e Oliveira, Fernanda Kelly2,3 (AUTHOR), Serraglio Fortes, Isadora1,6,7 (AUTHOR), Maciel Fernandes, Thaís Helena1,8 (AUTHOR), Barbosa da Silva, Elany1 (AUTHOR), Fajtova, Pavla1 (AUTHOR), Skinner, Danielle E.1 (AUTHOR), Syed, Rafay O.1 (AUTHOR), Lage de Siqueira-Neto, Jair1 (AUTHOR), Poso, Antti5,9 (AUTHOR), Fernandes Mota, Bruno Eduardo3 (AUTHOR), Alves Coelho-dos-Reis, Jordana Grazziela2 (AUTHOR), Santos Abrahão, Jônatas2 (AUTHOR), Gonçalves Maltarollo, Vinícius10 (AUTHOR), O'Donoghue, Anthony J.1 (AUTHOR) ajodonoghue@health.ucsd.edu, Caffrey, Conor R.1 (AUTHOR) ccaffrey@health.ucsd.edu
Source: Journal of Enzyme Inhibition & Medicinal Chemistry. Dec2025, Vol. 40 Issue 1, p1-24. 24p.
Database: Academic Search Ultimate
Full text is not displayed to guests.
FullText Links:
  – Type: pdflink
Text:
  Availability: 1
Header DbId: asn
DbLabel: Academic Search Ultimate
An: 190283313
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Discovery of benzyl carbamate inhibitors of coronavirus M<superscript>pro</superscript> enzymes from a legacy collection of cysteine protease inhibitors.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AR" term="%22Sá+Magalhães+Serafim%2C+Mateus%22">Sá Magalhães Serafim, Mateus</searchLink><relatesTo>1,2,3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Kronenberger%2C+Thales%22">Kronenberger, Thales</searchLink><relatesTo>4,5</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Francisco%2C+Karol+R%2E%22">Francisco, Karol R.</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22de+Sousa+Reis%2C+Erik+Vinicius%22">de Sousa Reis, Erik Vinicius</searchLink><relatesTo>2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Gonçalves+de+Oliveira%2C+Ellen%22">Gonçalves de Oliveira, Ellen</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Marcelino+e+Oliveira%2C+Fernanda+Kelly%22">Marcelino e Oliveira, Fernanda Kelly</searchLink><relatesTo>2,3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Serraglio+Fortes%2C+Isadora%22">Serraglio Fortes, Isadora</searchLink><relatesTo>1,6,7</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Maciel+Fernandes%2C+Thaís+Helena%22">Maciel Fernandes, Thaís Helena</searchLink><relatesTo>1,8</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Barbosa+da+Silva%2C+Elany%22">Barbosa da Silva, Elany</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Fajtova%2C+Pavla%22">Fajtova, Pavla</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Skinner%2C+Danielle+E%2E%22">Skinner, Danielle E.</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Syed%2C+Rafay+O%2E%22">Syed, Rafay O.</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Lage+de+Siqueira-Neto%2C+Jair%22">Lage de Siqueira-Neto, Jair</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Poso%2C+Antti%22">Poso, Antti</searchLink><relatesTo>5,9</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Fernandes+Mota%2C+Bruno+Eduardo%22">Fernandes Mota, Bruno Eduardo</searchLink><relatesTo>3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Alves+Coelho-dos-Reis%2C+Jordana+Grazziela%22">Alves Coelho-dos-Reis, Jordana Grazziela</searchLink><relatesTo>2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Santos+Abrahão%2C+Jônatas%22">Santos Abrahão, Jônatas</searchLink><relatesTo>2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Gonçalves+Maltarollo%2C+Vinícius%22">Gonçalves Maltarollo, Vinícius</searchLink><relatesTo>10</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22O'Donoghue%2C+Anthony+J%2E%22">O'Donoghue, Anthony J.</searchLink><relatesTo>1</relatesTo> (AUTHOR)<i> ajodonoghue@health.ucsd.edu</i><br /><searchLink fieldCode="AR" term="%22Caffrey%2C+Conor+R%2E%22">Caffrey, Conor R.</searchLink><relatesTo>1</relatesTo> (AUTHOR)<i> ccaffrey@health.ucsd.edu</i>
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%22Journal+of+Enzyme+Inhibition+%26+Medicinal+Chemistry%22">Journal of Enzyme Inhibition & Medicinal Chemistry</searchLink>. Dec2025, Vol. 40 Issue 1, p1-24. 24p.
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=190283313
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1080/14756366.2025.2585619
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        PageCount: 24
        StartPage: 1
    Titles:
      – TitleFull: Discovery of benzyl carbamate inhibitors of coronavirus Mpro enzymes from a legacy collection of cysteine protease inhibitors.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Sá Magalhães Serafim, Mateus
      – PersonEntity:
          Name:
            NameFull: Kronenberger, Thales
      – PersonEntity:
          Name:
            NameFull: Francisco, Karol R.
      – PersonEntity:
          Name:
            NameFull: de Sousa Reis, Erik Vinicius
      – PersonEntity:
          Name:
            NameFull: Gonçalves de Oliveira, Ellen
      – PersonEntity:
          Name:
            NameFull: Marcelino e Oliveira, Fernanda Kelly
      – PersonEntity:
          Name:
            NameFull: Serraglio Fortes, Isadora
      – PersonEntity:
          Name:
            NameFull: Maciel Fernandes, Thaís Helena
      – PersonEntity:
          Name:
            NameFull: Barbosa da Silva, Elany
      – PersonEntity:
          Name:
            NameFull: Fajtova, Pavla
      – PersonEntity:
          Name:
            NameFull: Skinner, Danielle E.
      – PersonEntity:
          Name:
            NameFull: Syed, Rafay O.
      – PersonEntity:
          Name:
            NameFull: Lage de Siqueira-Neto, Jair
      – PersonEntity:
          Name:
            NameFull: Poso, Antti
      – PersonEntity:
          Name:
            NameFull: Fernandes Mota, Bruno Eduardo
      – PersonEntity:
          Name:
            NameFull: Alves Coelho-dos-Reis, Jordana Grazziela
      – PersonEntity:
          Name:
            NameFull: Santos Abrahão, Jônatas
      – PersonEntity:
          Name:
            NameFull: Gonçalves Maltarollo, Vinícius
      – PersonEntity:
          Name:
            NameFull: O'Donoghue, Anthony J.
      – PersonEntity:
          Name:
            NameFull: Caffrey, Conor R.
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 01
              M: 12
              Text: Dec2025
              Type: published
              Y: 2025
          Identifiers:
            – Type: issn-print
              Value: 14756366
          Numbering:
            – Type: volume
              Value: 40
            – Type: issue
              Value: 1
          Titles:
            – TitleFull: Journal of Enzyme Inhibition & Medicinal Chemistry
              Type: main
ResultId 1