Ensuring enantiomeric consistency in FAPI radiopharmaceuticals: comparative analysis of (S)- and (S/R)-FAPI-46/-74 confirms pharmacological equivalence.

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Title: Ensuring enantiomeric consistency in FAPI radiopharmaceuticals: comparative analysis of (S)- and (S/R)-FAPI-46/-74 confirms pharmacological equivalence.
Authors: Staniszewska, Magdalena1 (AUTHOR) magdalena.staniszewska@uk-essen.de, Hübner, Ralph1 (AUTHOR) Ralph.Huebner@ext.uk-essen.de, Locatelli, Camilla1 (AUTHOR) camilla.locatelli@uk-essen.de, Howard, Douglas1 (AUTHOR) dougiehow2@gmail.com, Forni, Matilde2 (AUTHOR) Matilde.Forni@gehealthcare.com, Man, Francis3 (AUTHOR) Francis.Man@gehealthcare.com, Schoultz, Bent Wilhelm4 (AUTHOR) bent.wilhelm.schoultz@syklotronsenteret.no, Nuruddin, Syed4 (AUTHOR) Syed.Nuruddin@syklotronsenteret.no, Norberg-Schulz Hagen, Ingrid Sofie4 (AUTHOR) ingrid.hagen@syklotronsenteret.no, Mosessian, Sherly5 (AUTHOR) sherly.mosessian@sofie.com, Herrmann, Ken1 (AUTHOR) ken.herrmann@uk-essen.de, von Kiedrowski, Valeska1 (AUTHOR) valeska.vonkiedrowski@uk-essen.de, Lückerath, Katharina1 (AUTHOR) katharina.lueckerath@uk-essen.de
Source: EJNMMI Radiopharmacy & Chemistry. 2/28/2026, Vol. 11 Issue 1, p1-13. 13p.
Database: Academic Search Ultimate
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ISSN:2365421X
DOI:10.1186/s41181-026-00432-4