Targeting Steroid-Metabolizing Enzymes with 15β-Substituted Estrone Analogues: Dual Discovery of AKR1C2/17β-HSD1 Inhibitors and a Fluorescent 17β-HSD1 Ligand.
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| Title: | Targeting Steroid-Metabolizing Enzymes with 15β-Substituted Estrone Analogues: Dual Discovery of AKR1C2/17β-HSD1 Inhibitors and a Fluorescent 17β-HSD1 Ligand. |
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| Authors: | Resch, Vivien1 (AUTHOR), Gjorgoska, Marija2 (AUTHOR), Hafner, Eva2,3 (AUTHOR), Bacsa, Ildikó3,4 (AUTHOR), Kovács, Benjamin3,5 (AUTHOR), Büdefeld, Tomaž2,6 (AUTHOR), Hunyadi, Attila3,4,7 (AUTHOR), Huliák, Ildikó1,5 (AUTHOR), Kiricsi, Mónika2,5 (AUTHOR), Paragi, Gábor1,3,6,7 (AUTHOR), Rižner, Tea Lanišnik2,4 (AUTHOR), Mernyák, Erzsébet3,5 (AUTHOR) |
| Source: | Cancers. Jun2026, Vol. 18 Issue 12, p1889. 19p. |
| Database: | Academic Search Ultimate |
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| ISSN: | 20726694 |
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| DOI: | 10.3390/cancers18121889 |