Targeting Steroid-Metabolizing Enzymes with 15β-Substituted Estrone Analogues: Dual Discovery of AKR1C2/17β-HSD1 Inhibitors and a Fluorescent 17β-HSD1 Ligand.
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| Title: | Targeting Steroid-Metabolizing Enzymes with 15β-Substituted Estrone Analogues: Dual Discovery of AKR1C2/17β-HSD1 Inhibitors and a Fluorescent 17β-HSD1 Ligand. |
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| Authors: | Resch, Vivien1 (AUTHOR), Gjorgoska, Marija2 (AUTHOR), Hafner, Eva2,3 (AUTHOR), Bacsa, Ildikó3,4 (AUTHOR), Kovács, Benjamin3,5 (AUTHOR), Büdefeld, Tomaž2,6 (AUTHOR), Hunyadi, Attila3,4,7 (AUTHOR), Huliák, Ildikó1,5 (AUTHOR), Kiricsi, Mónika2,5 (AUTHOR), Paragi, Gábor1,3,6,7 (AUTHOR), Rižner, Tea Lanišnik2,4 (AUTHOR), Mernyák, Erzsébet3,5 (AUTHOR) |
| Source: | Cancers. Jun2026, Vol. 18 Issue 12, p1889. 19p. |
| Database: | Academic Search Ultimate |
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| FullText | Links: – Type: pdflink Text: Availability: 1 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 194911091 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Targeting Steroid-Metabolizing Enzymes with 15β-Substituted Estrone Analogues: Dual Discovery of AKR1C2/17β-HSD1 Inhibitors and a Fluorescent 17β-HSD1 Ligand. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AR" term="%22Resch%2C+Vivien%22">Resch, Vivien</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Gjorgoska%2C+Marija%22">Gjorgoska, Marija</searchLink><relatesTo>2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Hafner%2C+Eva%22">Hafner, Eva</searchLink><relatesTo>2,3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Bacsa%2C+Ildikó%22">Bacsa, Ildikó</searchLink><relatesTo>3,4</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Kovács%2C+Benjamin%22">Kovács, Benjamin</searchLink><relatesTo>3,5</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Büdefeld%2C+Tomaž%22">Büdefeld, Tomaž</searchLink><relatesTo>2,6</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Hunyadi%2C+Attila%22">Hunyadi, Attila</searchLink><relatesTo>3,4,7</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Huliák%2C+Ildikó%22">Huliák, Ildikó</searchLink><relatesTo>1,5</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Kiricsi%2C+Mónika%22">Kiricsi, Mónika</searchLink><relatesTo>2,5</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Paragi%2C+Gábor%22">Paragi, Gábor</searchLink><relatesTo>1,3,6,7</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Rižner%2C+Tea+Lanišnik%22">Rižner, Tea Lanišnik</searchLink><relatesTo>2,4</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Mernyák%2C+Erzsébet%22">Mernyák, Erzsébet</searchLink><relatesTo>3,5</relatesTo> (AUTHOR) – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22Cancers%22">Cancers</searchLink>. Jun2026, Vol. 18 Issue 12, p1889. 19p. |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=194911091 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.3390/cancers18121889 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 19 StartPage: 1889 Titles: – TitleFull: Targeting Steroid-Metabolizing Enzymes with 15β-Substituted Estrone Analogues: Dual Discovery of AKR1C2/17β-HSD1 Inhibitors and a Fluorescent 17β-HSD1 Ligand. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Resch, Vivien – PersonEntity: Name: NameFull: Gjorgoska, Marija – PersonEntity: Name: NameFull: Hafner, Eva – PersonEntity: Name: NameFull: Bacsa, Ildikó – PersonEntity: Name: NameFull: Kovács, Benjamin – PersonEntity: Name: NameFull: Büdefeld, Tomaž – PersonEntity: Name: NameFull: Hunyadi, Attila – PersonEntity: Name: NameFull: Huliák, Ildikó – PersonEntity: Name: NameFull: Kiricsi, Mónika – PersonEntity: Name: NameFull: Paragi, Gábor – PersonEntity: Name: NameFull: Rižner, Tea Lanišnik – PersonEntity: Name: NameFull: Mernyák, Erzsébet IsPartOfRelationships: – BibEntity: Dates: – D: 15 M: 06 Text: Jun2026 Type: published Y: 2026 Identifiers: – Type: issn-print Value: 20726694 Numbering: – Type: volume Value: 18 – Type: issue Value: 12 Titles: – TitleFull: Cancers Type: main |
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