Discovery of potent and orally bioavailable heterocycle-based cannabinoid CB1 receptor agonists

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Bibliographic Details
Title: Discovery of potent and orally bioavailable heterocycle-based cannabinoid CB1 receptor agonists
Authors: Kiyoi, Takao1, Adam, Julia M.1 juliaadam@blueyonder.co.uk, Clark, John K.1, Davies, Keneth1, Easson, Anna-Marie1, Edwards, Darren1, Feilden, Helen1, Fields, Ruth1, Francis, Stuart1, Jeremiah, Fiona1, McArthur, Duncan1, Morrison, Angus J.1, Prosser, Alan1, Ratcliffe, Paul D.1, Schulz, Jurgen1, Wishart, Grant1, Baker, James2, Campbell, Robert2, Cottney, Jean E.2, Deehan, Maureen2
Source: Bioorganic & Medicinal Chemistry Letters. Mar2011, Vol. 21 Issue 6, p1748-1753. 6p.
Database: Academic Search Ultimate
Description
ISSN:0960894X
DOI:10.1016/j.bmcl.2011.01.082