Design, synthesis and structure–activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate

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Bibliographic Details
Title: Design, synthesis and structure–activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate
Authors: Ratcliffe, Paul1 Paul.Ratcliffe@grunenthal.com, Adam, Julia M.1, Baker, James2, Bursi, Roberta3, Campbell, Robert2, Clark, John K.1, Cottney, Jean E.2, Deehan, Maureen2, Easson, Anna-Marie1, Ecker, Daniel4, Edwards, Darren1, Epemolu, Ola2, Evans, Louise2, Fields, Ruth1, Francis, Stuart1, Harradine, Paul1, Jeremiah, Fiona1, Kiyoi, Takao1, McArthur, Duncan1, Morrison, Angus1
Source: Bioorganic & Medicinal Chemistry Letters. Apr2011, Vol. 21 Issue 8, p2541-2546. 6p.
Database: Academic Search Ultimate
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