4-(3-Chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-methoxypyridin-2-yl)piperazine-1-carbothioamide(ML267), a Potent Inhibitor of Bacterial Phosphopantetheinyl TransferaseThat Attenuates Secondary Metabolism and Thwarts Bacterial Growth.

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Title: 4-(3-Chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-methoxypyridin-2-yl)piperazine-1-carbothioamide(ML267), a Potent Inhibitor of Bacterial Phosphopantetheinyl TransferaseThat Attenuates Secondary Metabolism and Thwarts Bacterial Growth.
Authors: Foley, Timothy L.1, Rai, Ganesha1, Yasgar, Adam1, Daniel, Thomas1, Baker, Heather L.1, Attene-Ramos, Matias1, Kosa, Nicolas M.1, Leister, William1, Burkart, Michael D.1, Jadhav, Ajit1, Simeonov, Anton1, Maloney, David J.1
Source: Journal of Medicinal Chemistry. Feb2014, Vol. 57 Issue 3, p1063-1078. 16p.
Database: Academic Search Ultimate
Description
ISSN:00222623
DOI:10.1021/jm401752p