Carfentanil stabilizes µ opioid receptor conformations that are ultra-efficient in inhibiting cAMP, resistant to naloxone or nalmefene but sensitive to naltrexone.

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Title: Carfentanil stabilizes µ opioid receptor conformations that are ultra-efficient in inhibiting cAMP, resistant to naloxone or nalmefene but sensitive to naltrexone.
Authors: Endt, Franziska1 (AUTHOR), Guo, Tao1 (AUTHOR), Steinritz, Dirk2 (AUTHOR), Amend, Niko2 (AUTHOR), Gudermann, Thomas1 (AUTHOR), Breit, Andreas1 (AUTHOR) andreas.breit@lrz.uni-muenchen.de
Source: Archives of Toxicology. Jul2025, Vol. 99 Issue 7, p2903-2915. 13p.
Database: Environment Complete
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ISSN:03405761
DOI:10.1007/s00204-025-04048-6