Pharmacological and pharmacokinetic properties of a structurally novel, potent, and selective metabotropic glutamate 2/3 receptor agonist: in vitro characterization of agonist (-)-(1R,4S,5S,6S)-4-amino-2-sulfonylbicyclo[3.1.0]-hexane-4,6-dicarboxylic acid (LY404039).

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Title: Pharmacological and pharmacokinetic properties of a structurally novel, potent, and selective metabotropic glutamate 2/3 receptor agonist: in vitro characterization of agonist (-)-(1R,4S,5S,6S)-4-amino-2-sulfonylbicyclo[3.1.0]-hexane-4,6-dicarboxylic acid (LY404039).
Authors: Rorick-Kehn LM; Neuroscience Discovery Research, Lilly Research Laboratories, Lilly Corporate Center, DC0510, Indianapolis, IN 46285, USA., Johnson BG, Burkey JL, Wright RA, Calligaro DO, Marek GJ, Nisenbaum ES, Catlow JT, Kingston AE, Giera DD, Herin MF, Monn JA, McKinzie DL, Schoepp DD
Source: The Journal of pharmacology and experimental therapeutics [J Pharmacol Exp Ther] 2007 Apr; Vol. 321 (1), pp. 308-17. Date of Electronic Publication: 2007 Jan 04.
Publication Type: Comparative Study; Journal Article
Journal Info: Publisher: Elsevier Country of Publication: Netherlands NLM ID: 0376362 Publication Model: Print-Electronic Cited Medium: Print ISSN: 0022-3565 (Print) Linking ISSN: 00223565 NLM ISO Abbreviation: J Pharmacol Exp Ther Subsets: MEDLINE
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  Data: Pharmacological and pharmacokinetic properties of a structurally novel, potent, and selective metabotropic glutamate 2/3 receptor agonist: in vitro characterization of agonist (-)-(1R,4S,5S,6S)-4-amino-2-sulfonylbicyclo[3.1.0]-hexane-4,6-dicarboxylic acid (LY404039).
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  Data: <searchLink fieldCode="AU" term="%22Rorick-Kehn+LM%22">Rorick-Kehn LM</searchLink>; Neuroscience Discovery Research, Lilly Research Laboratories, Lilly Corporate Center, DC0510, Indianapolis, IN 46285, USA.<br /><searchLink fieldCode="AU" term="%22Johnson+BG%22">Johnson BG</searchLink><br /><searchLink fieldCode="AU" term="%22Burkey+JL%22">Burkey JL</searchLink><br /><searchLink fieldCode="AU" term="%22Wright+RA%22">Wright RA</searchLink><br /><searchLink fieldCode="AU" term="%22Calligaro+DO%22">Calligaro DO</searchLink><br /><searchLink fieldCode="AU" term="%22Marek+GJ%22">Marek GJ</searchLink><br /><searchLink fieldCode="AU" term="%22Nisenbaum+ES%22">Nisenbaum ES</searchLink><br /><searchLink fieldCode="AU" term="%22Catlow+JT%22">Catlow JT</searchLink><br /><searchLink fieldCode="AU" term="%22Kingston+AE%22">Kingston AE</searchLink><br /><searchLink fieldCode="AU" term="%22Giera+DD%22">Giera DD</searchLink><br /><searchLink fieldCode="AU" term="%22Herin+MF%22">Herin MF</searchLink><br /><searchLink fieldCode="AU" term="%22Monn+JA%22">Monn JA</searchLink><br /><searchLink fieldCode="AU" term="%22McKinzie+DL%22">McKinzie DL</searchLink><br /><searchLink fieldCode="AU" term="%22Schoepp+DD%22">Schoepp DD</searchLink>
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier%22">Elsevier </searchLink><i>Country of Publication: </i>Netherlands <i>NLM ID: </i>0376362 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Print <i>ISSN: </i>0022-3565 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200223565%22">00223565 </searchLink><i>NLM ISO Abbreviation: </i>J Pharmacol Exp Ther <i>Subsets: </i>MEDLINE
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        Value: 10.1124/jpet.106.110809
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        StartPage: 308
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      – TitleFull: Pharmacological and pharmacokinetic properties of a structurally novel, potent, and selective metabotropic glutamate 2/3 receptor agonist: in vitro characterization of agonist (-)-(1R,4S,5S,6S)-4-amino-2-sulfonylbicyclo[3.1.0]-hexane-4,6-dicarboxylic acid (LY404039).
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              Text: 2007 Apr
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