Non-aromatic A-ring replacement in the triaryl bis-sulfone CB2 receptor inhibitors.
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| Title: | Non-aromatic A-ring replacement in the triaryl bis-sulfone CB2 receptor inhibitors. |
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| Authors: | Gilbert EJ; Department of Medicinal Chemistry, Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ 07033-0539, USA. eric.gilbert@spcorp.com, Zhou G, Wong MK, Tong L, Shankar BB, Huang C, Kelly J, Lavey BJ, McCombie SW, Chen L, Rizvi R, Dong Y, Shu Y, Kozlowski JA, Shih NY, Hipkin RW, Gonsiorek W, Malikzay A, Lunn CA, Favreau L, Lundell DJ |
| Source: | Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2010 Jan 15; Vol. 20 (2), pp. 608-11. Date of Electronic Publication: 2009 Nov 22. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 20005710 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Non-aromatic A-ring replacement in the triaryl bis-sulfone CB2 receptor inhibitors. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Gilbert+EJ%22">Gilbert EJ</searchLink>; Department of Medicinal Chemistry, Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ 07033-0539, USA. eric.gilbert@spcorp.com<br /><searchLink fieldCode="AU" term="%22Zhou+G%22">Zhou G</searchLink><br /><searchLink fieldCode="AU" term="%22Wong+MK%22">Wong MK</searchLink><br /><searchLink fieldCode="AU" term="%22Tong+L%22">Tong L</searchLink><br /><searchLink fieldCode="AU" term="%22Shankar+BB%22">Shankar BB</searchLink><br /><searchLink fieldCode="AU" term="%22Huang+C%22">Huang C</searchLink><br /><searchLink fieldCode="AU" term="%22Kelly+J%22">Kelly J</searchLink><br /><searchLink fieldCode="AU" term="%22Lavey+BJ%22">Lavey BJ</searchLink><br /><searchLink fieldCode="AU" term="%22McCombie+SW%22">McCombie SW</searchLink><br /><searchLink fieldCode="AU" term="%22Chen+L%22">Chen L</searchLink><br /><searchLink fieldCode="AU" term="%22Rizvi+R%22">Rizvi R</searchLink><br /><searchLink fieldCode="AU" term="%22Dong+Y%22">Dong Y</searchLink><br /><searchLink fieldCode="AU" term="%22Shu+Y%22">Shu Y</searchLink><br /><searchLink fieldCode="AU" term="%22Kozlowski+JA%22">Kozlowski JA</searchLink><br /><searchLink fieldCode="AU" term="%22Shih+NY%22">Shih NY</searchLink><br /><searchLink fieldCode="AU" term="%22Hipkin+RW%22">Hipkin RW</searchLink><br /><searchLink fieldCode="AU" term="%22Gonsiorek+W%22">Gonsiorek W</searchLink><br /><searchLink fieldCode="AU" term="%22Malikzay+A%22">Malikzay A</searchLink><br /><searchLink fieldCode="AU" term="%22Lunn+CA%22">Lunn CA</searchLink><br /><searchLink fieldCode="AU" term="%22Favreau+L%22">Favreau L</searchLink><br /><searchLink fieldCode="AU" term="%22Lundell+DJ%22">Lundell DJ</searchLink> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2010 Jan 15; Vol. 20 (2), pp. 608-11. <i>Date of Electronic Publication: </i>2009 Nov 22. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=20005710 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2009.11.084 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 608 Titles: – TitleFull: Non-aromatic A-ring replacement in the triaryl bis-sulfone CB2 receptor inhibitors. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Gilbert EJ – PersonEntity: Name: NameFull: Zhou G – PersonEntity: Name: NameFull: Wong MK – PersonEntity: Name: NameFull: Tong L – PersonEntity: Name: NameFull: Shankar BB – PersonEntity: Name: NameFull: Huang C – PersonEntity: Name: NameFull: Kelly J – PersonEntity: Name: NameFull: Lavey BJ – PersonEntity: Name: NameFull: McCombie SW – PersonEntity: Name: NameFull: Chen L – PersonEntity: Name: NameFull: Rizvi R – PersonEntity: Name: NameFull: Dong Y – PersonEntity: Name: NameFull: Shu Y – PersonEntity: Name: NameFull: Kozlowski JA – PersonEntity: Name: NameFull: Shih NY – PersonEntity: Name: NameFull: Hipkin RW – PersonEntity: Name: NameFull: Gonsiorek W – PersonEntity: Name: NameFull: Malikzay A – PersonEntity: Name: NameFull: Lunn CA – PersonEntity: Name: NameFull: Favreau L – PersonEntity: Name: NameFull: Lundell DJ IsPartOfRelationships: – BibEntity: Dates: – D: 15 M: 01 Text: 2010 Jan 15 Type: published Y: 2010 Identifiers: – Type: issn-electronic Value: 1464-3405 Numbering: – Type: volume Value: 20 – Type: issue Value: 2 Titles: – TitleFull: Bioorganic & medicinal chemistry letters Type: main |
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