Beyond small-molecule SAR: using the dopamine D3 receptor crystal structure to guide drug design.

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Title: Beyond small-molecule SAR: using the dopamine D3 receptor crystal structure to guide drug design.
Authors: Keck TM; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program, Baltimore, Maryland, USA., Burzynski C; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program, Baltimore, Maryland, USA., Shi L; Department of Physiology and Biophysics and Institute for Computational Biomedicine, Weill Cornell Medical College, New York, USA., Newman AH; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program, Baltimore, Maryland, USA. Electronic address: anewman@intra.nida.nih.gov.
Source: Advances in pharmacology (San Diego, Calif.) [Adv Pharmacol] 2014; Vol. 69, pp. 267-300.
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Review
Journal Info: Publisher: Academic Press Country of Publication: United States NLM ID: 9015397 Publication Model: Print Cited Medium: Internet ISSN: 1557-8925 (Electronic) Linking ISSN: 10543589 NLM ISO Abbreviation: Adv Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: <searchLink fieldCode="AU" term="%22Keck+TM%22">Keck TM</searchLink>; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program, Baltimore, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Burzynski+C%22">Burzynski C</searchLink>; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program, Baltimore, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Shi+L%22">Shi L</searchLink>; Department of Physiology and Biophysics and Institute for Computational Biomedicine, Weill Cornell Medical College, New York, USA.<br /><searchLink fieldCode="AU" term="%22Newman+AH%22">Newman AH</searchLink>; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program, Baltimore, Maryland, USA. Electronic address: anewman@intra.nida.nih.gov.
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        Value: 10.1016/B978-0-12-420118-7.00007-X
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      – Code: eng
        Text: English
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              Text: 2014
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              Value: 69
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