Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists.

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Title: Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists.
Authors: Hintermann S; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Guntermann C; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Mattes H; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Carcache DA; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Wagner J; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Vulpetti A; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Billich A; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Dawson J; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Kaupmann K; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Kallen J; CPC, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Stringer R; MAP, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Orain D; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.
Source: ChemMedChem [ChemMedChem] 2016 Dec 16; Vol. 11 (24), pp. 2640-2648. Date of Electronic Publication: 2016 Nov 30.
Publication Type: Journal Article
Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1860-7187
DOI:10.1002/cmdc.201600500