Investigation of piperazine benzamides as human β3 adrenergic receptor agonists for the treatment of overactive bladder.

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Title: Investigation of piperazine benzamides as human β3 adrenergic receptor agonists for the treatment of overactive bladder.
Authors: Harper BH; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States. Electronic address: bart_harper@merck.com., Wang L; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Zhu C; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Kar NF; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Li B; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Moyes CR; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Goble SD; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Costa M; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Dingley K; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Di Salvo J; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Ha SN; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Hurley A; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Li X; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Miller RR; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Nagabukuro H; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Salituro GM; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Smith S; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Struthers M; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Hale JJ; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Edmondson SD; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Berger R; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2017 Feb 15; Vol. 27 (4), pp. 1094-1098. Date of Electronic Publication: 2016 Dec 11.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Investigation of piperazine benzamides as human β<subscript>3</subscript> adrenergic receptor agonists for the treatment of overactive bladder.
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  Data: <searchLink fieldCode="AU" term="%22Harper+BH%22">Harper BH</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States. Electronic address: bart_harper@merck.com.<br /><searchLink fieldCode="AU" term="%22Wang+L%22">Wang L</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Zhu+C%22">Zhu C</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Kar+NF%22">Kar NF</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Li+B%22">Li B</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Moyes+CR%22">Moyes CR</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Goble+SD%22">Goble SD</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Costa+M%22">Costa M</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Dingley+K%22">Dingley K</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Di+Salvo+J%22">Di Salvo J</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Ha+SN%22">Ha SN</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Hurley+A%22">Hurley A</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Li+X%22">Li X</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Miller+RR%22">Miller RR</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Nagabukuro+H%22">Nagabukuro H</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Salituro+GM%22">Salituro GM</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Smith+S%22">Smith S</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Struthers+M%22">Struthers M</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Hale+JJ%22">Hale JJ</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Edmondson+SD%22">Edmondson SD</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Berger+R%22">Berger R</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.
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