Investigation of piperazine benzamides as human β3 adrenergic receptor agonists for the treatment of overactive bladder.
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| Title: | Investigation of piperazine benzamides as human β |
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| Authors: | Harper BH; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States. Electronic address: bart_harper@merck.com., Wang L; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Zhu C; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Kar NF; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Li B; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Moyes CR; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Goble SD; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Costa M; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Dingley K; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Di Salvo J; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Ha SN; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Hurley A; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Li X; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Miller RR; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Nagabukuro H; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Salituro GM; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Smith S; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Struthers M; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Hale JJ; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Edmondson SD; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Berger R; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States. |
| Source: | Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2017 Feb 15; Vol. 27 (4), pp. 1094-1098. Date of Electronic Publication: 2016 Dec 11. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 28089699 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Investigation of piperazine benzamides as human β<subscript>3</subscript> adrenergic receptor agonists for the treatment of overactive bladder. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Harper+BH%22">Harper BH</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States. Electronic address: bart&#95;harper@merck.com.<br /><searchLink fieldCode="AU" term="%22Wang+L%22">Wang L</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Zhu+C%22">Zhu C</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Kar+NF%22">Kar NF</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Li+B%22">Li B</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Moyes+CR%22">Moyes CR</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Goble+SD%22">Goble SD</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Costa+M%22">Costa M</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Dingley+K%22">Dingley K</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Di+Salvo+J%22">Di Salvo J</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Ha+SN%22">Ha SN</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Hurley+A%22">Hurley A</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Li+X%22">Li X</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Miller+RR%22">Miller RR</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Nagabukuro+H%22">Nagabukuro H</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Salituro+GM%22">Salituro GM</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Smith+S%22">Smith S</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Struthers+M%22">Struthers M</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Hale+JJ%22">Hale JJ</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Edmondson+SD%22">Edmondson SD</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.<br /><searchLink fieldCode="AU" term="%22Berger+R%22">Berger R</searchLink>; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2017 Feb 15; Vol. 27 (4), pp. 1094-1098. <i>Date of Electronic Publication: </i>2016 Dec 11. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=28089699 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2016.12.033 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 1094 Titles: – TitleFull: Investigation of piperazine benzamides as human β3 adrenergic receptor agonists for the treatment of overactive bladder. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Harper BH – PersonEntity: Name: NameFull: Wang L – PersonEntity: Name: NameFull: Zhu C – PersonEntity: Name: NameFull: Kar NF – PersonEntity: Name: NameFull: Li B – PersonEntity: Name: NameFull: Moyes CR – PersonEntity: Name: NameFull: Goble SD – PersonEntity: Name: NameFull: Costa M – PersonEntity: Name: NameFull: Dingley K – PersonEntity: Name: NameFull: Di Salvo J – PersonEntity: Name: NameFull: Ha SN – PersonEntity: Name: NameFull: Hurley A – PersonEntity: Name: NameFull: Li X – PersonEntity: Name: NameFull: Miller RR – PersonEntity: Name: NameFull: Nagabukuro H – PersonEntity: Name: NameFull: Salituro GM – PersonEntity: Name: NameFull: Smith S – PersonEntity: Name: NameFull: Struthers M – PersonEntity: Name: NameFull: Hale JJ – PersonEntity: Name: NameFull: Edmondson SD – PersonEntity: Name: NameFull: Berger R IsPartOfRelationships: – BibEntity: Dates: – D: 15 M: 02 Text: 2017 Feb 15 Type: published Y: 2017 Identifiers: – Type: issn-electronic Value: 1464-3405 Numbering: – Type: volume Value: 27 – Type: issue Value: 4 Titles: – TitleFull: Bioorganic & medicinal chemistry letters Type: main |
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