View in EDS

Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis.

Saved in:
Bibliographic Details
Title: Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis.
Authors: Thakkar M; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: mahesh.thakkar@advinus.com., Bhuniya D; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: debnath.bhuniya@advinus.com., Kaduskar R; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: rahul.kaduskar@advinus.com., Mengawade T; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: tanaji.m@advinus.com., Naik K; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: keshav.naik@advinus.com., Salunkhe V; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: videsh.salunkhe@advinus.com., Bhalerao A; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: amit.bhalerao@advinus.com., Kurhade S; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: santosh.kurhade@advinus.com., Mavinahalli J; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: jagadeesh.m@advinus.com., Jain V; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: vaibhav.jain@advinus.com., Petla R; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: rajkanth.petla@advinus.com., Avaragolla S; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: satheesh.a@advinus.com., Ray S; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: swagatam.ray@advinus.com., Rouduri S; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: sreekanth.r@advinus.com., Dhanave A; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: avinash.dhanave@advinus.com., De S; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: siddhartha.de@advinus.com., Pathade V; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: vishal.pathade@advinus.com., Tambe A; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: ashwini.tambe@advinus.com., Raje AA; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: amol.raje@advinus.com., Madgula V; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: vamsi.m@advinus.com., Joshi S; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: sachin.joshi@advinus.com., Nadeem A; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: ahmed.nadeem@advinus.com., Bala M; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: madhu.bala@advinus.com., Umrani D; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: dhananjay.umrani@advinus.com., Hariharan N; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: hariharan.narayanan@advinus.com., Kulkarni B; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: kulkarni.b@advinus.com., Mookhtiar KA; Drug Discovery Unit, Advinus Therapeutics Ltd, Plot-9, Phase-I, Rajiv Gandhi InfoTech Park, Hinjewadi, Pune 411057, India. Electronic address: kasim.mookhtiar@advinus.com.
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2017 Apr 15; Vol. 27 (8), pp. 1867-1873. Date of Electronic Publication: 2017 Feb 22.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1464-3405
DOI:10.1016/j.bmcl.2017.02.026