Effects of Drug-Antibody Ratio on Pharmacokinetics, Biodistribution, Efficacy, and Tolerability of Antibody-Maytansinoid Conjugates.

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Title: Effects of Drug-Antibody Ratio on Pharmacokinetics, Biodistribution, Efficacy, and Tolerability of Antibody-Maytansinoid Conjugates.
Authors: Sun X; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Ponte JF; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Yoder NC; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Laleau R; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Coccia J; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Lanieri L; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Qiu Q; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Wu R; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Hong E; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Bogalhas M; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Wang L; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Dong L; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Setiady Y; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Maloney EK; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Ab O; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Zhang X; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Pinkas J; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Keating TA; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Chari R; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Erickson HK; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States., Lambert JM; ImmunoGen, Inc. , 830 Winter Street, Waltham, Massachusetts 02451, United States.
Source: Bioconjugate chemistry [Bioconjug Chem] 2017 May 17; Vol. 28 (5), pp. 1371-1381. Date of Electronic Publication: 2017 Apr 13.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9010319 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4812 (Electronic) Linking ISSN: 10431802 NLM ISO Abbreviation: Bioconjug Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4812
DOI:10.1021/acs.bioconjchem.7b00062