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Azetidine and Piperidine Carbamates as Efficient, Covalent Inhibitors of Monoacylglycerol Lipase.

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Title: Azetidine and Piperidine Carbamates as Efficient, Covalent Inhibitors of Monoacylglycerol Lipase.
Authors: Butler CR; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States., Beck EM; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States., Harris A; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Huang Z; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States., McAllister LA; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States., Am Ende CW; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Fennell K; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Foley TL; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Fonseca K; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States., Hawrylik SJ; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Johnson DS; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States., Knafels JD; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Mente S; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States., Noell GS; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Pandit J; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Phillips TB; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Piro JR; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States., Rogers BN; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States., Samad TA; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States., Wang J; WuXi AppTec , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China., Wan S; WuXi AppTec , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China., Brodney MA; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2017 Dec 14; Vol. 60 (23), pp. 9860-9873. Date of Electronic Publication: 2017 Dec 05.
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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PubType: Academic Journal
PubTypeId: academicJournal
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  Data: Azetidine and Piperidine Carbamates as Efficient, Covalent Inhibitors of Monoacylglycerol Lipase.
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  Data: <searchLink fieldCode="AU" term="%22Butler+CR%22">Butler CR</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Beck+EM%22">Beck EM</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Harris+A%22">Harris A</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Huang+Z%22">Huang Z</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22McAllister+LA%22">McAllister LA</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Am+Ende+CW%22">Am Ende CW</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Fennell+K%22">Fennell K</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Foley+TL%22">Foley TL</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Fonseca+K%22">Fonseca K</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Hawrylik+SJ%22">Hawrylik SJ</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Johnson+DS%22">Johnson DS</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Knafels+JD%22">Knafels JD</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Mente+S%22">Mente S</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Noell+GS%22">Noell GS</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Pandit+J%22">Pandit J</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Phillips+TB%22">Phillips TB</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Piro+JR%22">Piro JR</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Rogers+BN%22">Rogers BN</searchLink>; Pfizer Worldwide Research and Development , 445 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Samad+TA%22">Samad TA</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Wang+J%22">Wang J</searchLink>; WuXi AppTec , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China.<br /><searchLink fieldCode="AU" term="%22Wan+S%22">Wan S</searchLink>; WuXi AppTec , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China.<br /><searchLink fieldCode="AU" term="%22Brodney+MA%22">Brodney MA</searchLink>; Pfizer Worldwide Research and Development , 1 Portland Street, Cambridge, Massachusetts 02139, United States.
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  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2017 Dec 14; Vol. 60 (23), pp. 9860-9873. <i>Date of Electronic Publication: </i>2017 Dec 05.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE
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        Value: 10.1021/acs.jmedchem.7b01531
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        Text: English
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              Text: 2017 Dec 14
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