Chemical Instability and Promiscuity of Arylmethylidenepyrazolinone-Based MDMX Inhibitors.

Saved in:
Bibliographic Details
Title: Chemical Instability and Promiscuity of Arylmethylidenepyrazolinone-Based MDMX Inhibitors.
Authors: Stefaniak J; Structural Genomics Consortium, Nuffield Department of Medicine , University of Oxford , Oxford , United Kingdom.; Target Discovery Institute, Nuffield Department of Medicine , University of Oxford , Oxford , United Kingdom.; Department of Chemistry, Chemistry Research Laboratory , University of Oxford , Oxford , United Kingdom., Lewis AM; Structural Genomics Consortium, Nuffield Department of Medicine , University of Oxford , Oxford , United Kingdom.; Target Discovery Institute, Nuffield Department of Medicine , University of Oxford , Oxford , United Kingdom., Conole D; Department of Chemistry, Chemistry Research Laboratory , University of Oxford , Oxford , United Kingdom., Galan SRG; Department of Chemistry, Chemistry Research Laboratory , University of Oxford , Oxford , United Kingdom., Bataille CJR; Department of Chemistry, Chemistry Research Laboratory , University of Oxford , Oxford , United Kingdom., Wynne GM; Department of Chemistry, Chemistry Research Laboratory , University of Oxford , Oxford , United Kingdom.; Department of Pharmacology , University of Oxford , Oxford , United Kingdom., Castaldi MP; Discovery Sciences, IMED Biotech Unit , AstraZeneca , Waltham , Massachusetts 02451 , United States., Lundbäck T; Discovery Sciences, IMED Biotech Unit , AstraZeneca , Gothenburg , Sweden., Russell AJ; Department of Chemistry, Chemistry Research Laboratory , University of Oxford , Oxford , United Kingdom.; Department of Pharmacology , University of Oxford , Oxford , United Kingdom., Huber KVM; Structural Genomics Consortium, Nuffield Department of Medicine , University of Oxford , Oxford , United Kingdom.; Target Discovery Institute, Nuffield Department of Medicine , University of Oxford , Oxford , United Kingdom.
Source: ACS chemical biology [ACS Chem Biol] 2018 Oct 19; Vol. 13 (10), pp. 2849-2854. Date of Electronic Publication: 2018 Sep 19.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1554-8937
DOI:10.1021/acschembio.8b00665