6-Phenylpyrimidin-4-ones as Positive Allosteric Modulators at the M1 mAChR: The Determinants of Allosteric Activity.
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| Title: | 6-Phenylpyrimidin-4-ones as Positive Allosteric Modulators at the M |
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| Authors: | Jörg M, van der Westhuizen ET, Khajehali E, Burger WAC, White JM; Bio21 Molecular Science and Biotechnology Institute , The University of Melbourne , 30 Flemington Road , Parkville 3010 , VIC , Australia., Choy KHC, Tobin AB; Centre for Translational Pharmacology, Institute of Molecular, Cell and Systems Biology, College of Medical, Veterinary and Life Sciences , University of Glasgow , Glasgow G12 8QQ , United Kingdom., Sexton PM, Valant C, Capuano B, Christopoulos A, Scammells PJ |
| Source: | ACS chemical neuroscience [ACS Chem Neurosci] 2019 Mar 20; Vol. 10 (3), pp. 1099-1114. Date of Electronic Publication: 2018 Dec 28. |
| Publication Type: | Journal Article; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101525337 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1948-7193 (Electronic) Linking ISSN: 19487193 NLM ISO Abbreviation: ACS Chem Neurosci Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| ISSN: | 1948-7193 |
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| DOI: | 10.1021/acschemneuro.8b00613 |