6-Phenylpyrimidin-4-ones as Positive Allosteric Modulators at the M1 mAChR: The Determinants of Allosteric Activity.
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| Title: | 6-Phenylpyrimidin-4-ones as Positive Allosteric Modulators at the M |
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| Authors: | Jörg M, van der Westhuizen ET, Khajehali E, Burger WAC, White JM; Bio21 Molecular Science and Biotechnology Institute , The University of Melbourne , 30 Flemington Road , Parkville 3010 , VIC , Australia., Choy KHC, Tobin AB; Centre for Translational Pharmacology, Institute of Molecular, Cell and Systems Biology, College of Medical, Veterinary and Life Sciences , University of Glasgow , Glasgow G12 8QQ , United Kingdom., Sexton PM, Valant C, Capuano B, Christopoulos A, Scammells PJ |
| Source: | ACS chemical neuroscience [ACS Chem Neurosci] 2019 Mar 20; Vol. 10 (3), pp. 1099-1114. Date of Electronic Publication: 2018 Dec 28. |
| Publication Type: | Journal Article; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101525337 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1948-7193 (Electronic) Linking ISSN: 19487193 NLM ISO Abbreviation: ACS Chem Neurosci Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 30547573 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: 6-Phenylpyrimidin-4-ones as Positive Allosteric Modulators at the M<subscript>1</subscript> mAChR: The Determinants of Allosteric Activity. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Jörg+M%22">Jörg M</searchLink><br /><searchLink fieldCode="AU" term="%22van+der+Westhuizen+ET%22">van der Westhuizen ET</searchLink><br /><searchLink fieldCode="AU" term="%22Khajehali+E%22">Khajehali E</searchLink><br /><searchLink fieldCode="AU" term="%22Burger+WAC%22">Burger WAC</searchLink><br /><searchLink fieldCode="AU" term="%22White+JM%22">White JM</searchLink>; Bio21 Molecular Science and Biotechnology Institute , The University of Melbourne , 30 Flemington Road , Parkville 3010 , VIC , Australia.<br /><searchLink fieldCode="AU" term="%22Choy+KHC%22">Choy KHC</searchLink><br /><searchLink fieldCode="AU" term="%22Tobin+AB%22">Tobin AB</searchLink>; Centre for Translational Pharmacology, Institute of Molecular, Cell and Systems Biology, College of Medical, Veterinary and Life Sciences , University of Glasgow , Glasgow G12 8QQ , United Kingdom.<br /><searchLink fieldCode="AU" term="%22Sexton+PM%22">Sexton PM</searchLink><br /><searchLink fieldCode="AU" term="%22Valant+C%22">Valant C</searchLink><br /><searchLink fieldCode="AU" term="%22Capuano+B%22">Capuano B</searchLink><br /><searchLink fieldCode="AU" term="%22Christopoulos+A%22">Christopoulos A</searchLink><br /><searchLink fieldCode="AU" term="%22Scammells+PJ%22">Scammells PJ</searchLink> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101525337%22">ACS chemical neuroscience</searchLink> [ACS Chem Neurosci] 2019 Mar 20; Vol. 10 (3), pp. 1099-1114. <i>Date of Electronic Publication: </i>2018 Dec 28. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Research Support, Non-U.S. Gov't – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101525337 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1948-7193 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219487193%22">19487193 </searchLink><i>NLM ISO Abbreviation: </i>ACS Chem Neurosci <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=30547573 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acschemneuro.8b00613 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 1099 Titles: – TitleFull: 6-Phenylpyrimidin-4-ones as Positive Allosteric Modulators at the M1 mAChR: The Determinants of Allosteric Activity. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Jörg M – PersonEntity: Name: NameFull: van der Westhuizen ET – PersonEntity: Name: NameFull: Khajehali E – PersonEntity: Name: NameFull: Burger WAC – PersonEntity: Name: NameFull: White JM – PersonEntity: Name: NameFull: Choy KHC – PersonEntity: Name: NameFull: Tobin AB – PersonEntity: Name: NameFull: Sexton PM – PersonEntity: Name: NameFull: Valant C – PersonEntity: Name: NameFull: Capuano B – PersonEntity: Name: NameFull: Christopoulos A – PersonEntity: Name: NameFull: Scammells PJ IsPartOfRelationships: – BibEntity: Dates: – D: 20 M: 03 Text: 2019 Mar 20 Type: published Y: 2019 Identifiers: – Type: issn-electronic Value: 1948-7193 Numbering: – Type: volume Value: 10 – Type: issue Value: 3 Titles: – TitleFull: ACS chemical neuroscience Type: main |
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