Bifunctional Duocarmycin Analogues as Inhibitors of Protein Tyrosine Kinases.

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Title: Bifunctional Duocarmycin Analogues as Inhibitors of Protein Tyrosine Kinases.
Authors: De Ford C; Department of Pharmaceutical Biology and Biotechnology , Albert Ludwigs University Freiburg , Stefan-Meier-Strasse 19 , D-79104 Freiburg , Germany.; Spemann Graduate School of Biology and Medicine (SGBM) , Albert Ludwigs University Freiburg , Albertstrasse 19a , 79104 Freiburg , Germany., Penchalaiah K; Institute of Organic and Biomolecular Chemistry , Georg-August University , Tammannstrasse 2 , 37077 Göttingen , Germany., Kreft A; Institute of Organic and Biomolecular Chemistry , Georg-August University , Tammannstrasse 2 , 37077 Göttingen , Germany., Humar M; Department of Pharmaceutical Biology and Biotechnology , Albert Ludwigs University Freiburg , Stefan-Meier-Strasse 19 , D-79104 Freiburg , Germany., Heydenreuter W; Institute of Organic Chemistry II , Technische Universität München , Lichtenbergstrasse 4 , 85747 Garching , Germany., Kangani M; Institute of Organic and Biomolecular Chemistry , Georg-August University , Tammannstrasse 2 , 37077 Göttingen , Germany., Sieber SA; Institute of Organic Chemistry II , Technische Universität München , Lichtenbergstrasse 4 , 85747 Garching , Germany., Tietze LF; Institute of Organic and Biomolecular Chemistry , Georg-August University , Tammannstrasse 2 , 37077 Göttingen , Germany., Merfort I; Department of Pharmaceutical Biology and Biotechnology , Albert Ludwigs University Freiburg , Stefan-Meier-Strasse 19 , D-79104 Freiburg , Germany.; Spemann Graduate School of Biology and Medicine (SGBM) , Albert Ludwigs University Freiburg , Albertstrasse 19a , 79104 Freiburg , Germany.
Source: Journal of natural products [J Nat Prod] 2019 Jan 25; Vol. 82 (1), pp. 16-26. Date of Electronic Publication: 2019 Jan 08.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Society of Pharmacognosy Country of Publication: United States NLM ID: 7906882 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-6025 (Electronic) Linking ISSN: 01633864 NLM ISO Abbreviation: J Nat Prod Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-6025
DOI:10.1021/acs.jnatprod.8b00233