Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity.

Saved in:
Bibliographic Details
Title: Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity.
Authors: Botros SS; Pharmacology Department, Theodor Bilharz Research Institute, Warrak El-Hadar, Imbaba, P.O. Box 30, Giza, 12411, Egypt., William S; Parasitology Department, Theodor Bilharz Research Institute, Warrak El-Hadar, Imbaba, P.O. Box 30, Giza, 12411, Egypt., Sabra AA; Pharmacology Department, Theodor Bilharz Research Institute, Warrak El-Hadar, Imbaba, P.O. Box 30, Giza, 12411, Egypt., El-Lakkany NM; Pharmacology Department, Theodor Bilharz Research Institute, Warrak El-Hadar, Imbaba, P.O. Box 30, Giza, 12411, Egypt., Seif El-Din SH; Pharmacology Department, Theodor Bilharz Research Institute, Warrak El-Hadar, Imbaba, P.O. Box 30, Giza, 12411, Egypt., García-Rubia A; Centro de Investigaciones Biológicas (CIB-CSIC), Madrid, Spain., Sebastián-Pérez V; Centro de Investigaciones Biológicas (CIB-CSIC), Madrid, Spain., Blaazer AR; Medicinal Chemistry Vrije Universiteit Amsterdam (VUA), the Netherlands., de Heuvel E; Medicinal Chemistry Vrije Universiteit Amsterdam (VUA), the Netherlands., Sijm M; Medicinal Chemistry Vrije Universiteit Amsterdam (VUA), the Netherlands., Zheng Y; Medicinal Chemistry Vrije Universiteit Amsterdam (VUA), the Netherlands., Salado IG; University of Antwerp (UA), Belgium., Munday JC; Institute of Infection, Immunity and Inflammation, University of Glasgow, Glasgow, G12 8TA, UK., Maes L; University of Antwerp (UA), Belgium., de Esch IJP; Medicinal Chemistry Vrije Universiteit Amsterdam (VUA), the Netherlands., Sterk GJ; Medicinal Chemistry Vrije Universiteit Amsterdam (VUA), the Netherlands., Augustyns K; University of Antwerp (UA), Belgium., Leurs R; Medicinal Chemistry Vrije Universiteit Amsterdam (VUA), the Netherlands., Gil C; Centro de Investigaciones Biológicas (CIB-CSIC), Madrid, Spain., De Koning HP; Institute of Infection, Immunity and Inflammation, University of Glasgow, Glasgow, G12 8TA, UK. Electronic address: Harry.de-Koning@glasgow.ac.uk.
Source: International journal for parasitology. Drugs and drug resistance [Int J Parasitol Drugs Drug Resist] 2019 Apr; Vol. 9, pp. 35-43. Date of Electronic Publication: 2019 Jan 14.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Elsevier Country of Publication: Netherlands NLM ID: 101576715 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2211-3207 (Electronic) Linking ISSN: 22113207 NLM ISO Abbreviation: Int J Parasitol Drugs Drug Resist Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2211-3207
DOI:10.1016/j.ijpddr.2019.01.001