Discovery of Novel µ-Opioid Receptor Inverse Agonist from a Combinatorial Library of Tetrapeptides through Structure-Based Virtual Screening.

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Title: Discovery of Novel µ-Opioid Receptor Inverse Agonist from a Combinatorial Library of Tetrapeptides through Structure-Based Virtual Screening.
Authors: Poli G; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126 Pisa, Italy., Dimmito MP; Department of Pharmacy, University of Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, 66100 Chieti, Italy., Mollica A; Department of Pharmacy, University of Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, 66100 Chieti, Italy., Zengin G; Department of Biology, Science Faculty, Selcuk University, 42130 Konya, Turkey., Benyhe S; Institute of Biochemistry, Biological Research Center, Hungarian Academy of Sciences, H-6726 Szeged, Temesvári krt. 62, 6726, Szeged, Hungary., Zador F; Institute of Biochemistry, Biological Research Center, Hungarian Academy of Sciences, H-6726 Szeged, Temesvári krt. 62, 6726, Szeged, Hungary., Stefanucci A; Department of Pharmacy, University of Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, 66100 Chieti, Italy.
Source: Molecules (Basel, Switzerland) [Molecules] 2019 Oct 27; Vol. 24 (21). Date of Electronic Publication: 2019 Oct 27.
Publication Type: Journal Article
Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049 (Electronic) Linking ISSN: 14203049 NLM ISO Abbreviation: Molecules Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1420-3049
DOI:10.3390/molecules24213872