Cellular Target Engagement Approaches to Monitor Epigenetic Reader Domain Interactions.

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Title: Cellular Target Engagement Approaches to Monitor Epigenetic Reader Domain Interactions.
Authors: Phillipou AN; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Lay CS; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Carver CE; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Messenger C; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Evans JP; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Lewis AJ; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Gordon LJ; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Mahmood M; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Greenhough LA; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Sammon D; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Cheng AT; Functional Genomics, Medicinal Science and Technology, GlaxoSmithKline, Collegeville, PA, USA., Chakraborty S; Functional Genomics, Medicinal Science and Technology, GlaxoSmithKline, Collegeville, PA, USA., Jones EJ; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Lucas SCC; Epigenetics Research Unit, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Gatfield KM; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Brierley DJ; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK., Craggs PD; Medicine Design, Medicinal Science and Technology, GlaxoSmithKline, Stevenage, Hertfordshire, UK.
Source: SLAS discovery : advancing life sciences R & D [SLAS Discov] 2020 Feb; Vol. 25 (2), pp. 163-175. Date of Electronic Publication: 2019 Dec 25.
Publication Type: Journal Article
Journal Info: Publisher: SAGE Publications Country of Publication: United States NLM ID: 101697563 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2472-5560 (Electronic) Linking ISSN: 24725552 NLM ISO Abbreviation: SLAS Discov Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2472-5560
DOI:10.1177/2472555219896278