Intestinal P-gp and Putative Hepatic OATP1B Induction: International Transporter Consortium Perspective on Drug Development Implications.
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| Title: | Intestinal P-gp and Putative Hepatic OATP1B Induction: International Transporter Consortium Perspective on Drug Development Implications. |
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| Authors: | Zamek-Gliszczynski MJ; Drug Meabolism and Pharmacokinetics, GlaxoSmithKline, Collegeville, Pennsylvania, USA., Patel M; Pharmacokinetics and Drug Metabolism, Amgen Research, Cambridge, Massachusetts, USA., Yang X; Office of Clinical Pharmacology, US Food and Drug Administration, Silver Spring, Maryland, USA., Lutz JD; Department of Clinical Pharmacology, Gilead Sciences, Inc, Foster City, California, USA., Chu X; Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & CO., Inc, Kenilworth, New Jersey, USA., Brouwer KLR; Division of Pharmacotherapy and Experimental Therapeutics, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA., Lai Y; Drug Metabolism, Gilead Sciences, Inc., Foster City, California, USA., Lee CA; Nonclinical Development and Clinical Pharmacology, Arena Pharmaceuticals, San Diego, California, USA., Neuhoff S; Simcyp Division, Certara UK Limited, Sheffield, UK., Paine MF; Department of Pharmaceutical Sciences, College of Pharmacy and Pharmaceutical Sciences, Washington State University, Spokane, Washington, USA., Sugiyama Y; Sugiyama Laboratory, RIKEN Baton Zone, Program, RIKEN Cluster for Science, RIKEN, Yokohama, Kanagawa, Japan., Taskar KS; Drug Meabolism and Pharmacokinetics, GlaxoSmithKline, Ware, UK., Galetin A; Centre for Applied Pharmacokinetic Research, School of Health Sciences, The University of Manchester, Manchester, UK. |
| Source: | Clinical pharmacology and therapeutics [Clin Pharmacol Ther] 2021 Jan; Vol. 109 (1), pp. 55-64. Date of Electronic Publication: 2020 Jul 09. |
| Publication Type: | Journal Article; Research Support, N.I.H., Extramural; Review |
| Journal Info: | Publisher: Wiley Country of Publication: United States NLM ID: 0372741 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1532-6535 (Electronic) Linking ISSN: 00099236 NLM ISO Abbreviation: Clin Pharmacol Ther Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| ISSN: | 1532-6535 |
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| DOI: | 10.1002/cpt.1916 |