High Throughput Screen Identifies the DNMT1 (DNA Methyltransferase-1) Inhibitor, 5-Azacytidine, as a Potent Inducer of PTEN (Phosphatase and Tensin Homolog): Central Role for PTEN in 5-Azacytidine Protection Against Pathological Vascular Remodeling.

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Title: High Throughput Screen Identifies the DNMT1 (DNA Methyltransferase-1) Inhibitor, 5-Azacytidine, as a Potent Inducer of PTEN (Phosphatase and Tensin Homolog): Central Role for PTEN in 5-Azacytidine Protection Against Pathological Vascular Remodeling.
Authors: Strand KA; From the Division of Renal Diseases and Hypertension, Department of Medicine (K.A.S., S.L., M.F.M., A.J.J., A.M.D., R.A.N., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora., Lu S; From the Division of Renal Diseases and Hypertension, Department of Medicine (K.A.S., S.L., M.F.M., A.J.J., A.M.D., R.A.N., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora., Mutryn MF; From the Division of Renal Diseases and Hypertension, Department of Medicine (K.A.S., S.L., M.F.M., A.J.J., A.M.D., R.A.N., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora., Li L; School of Pharmacy and Pharmaceutical Sciences (L.L., Q.Z., D.V.L.), University of Colorado, Anschutz Medical Campus, Aurora., Zhou Q; School of Pharmacy and Pharmaceutical Sciences (L.L., Q.Z., D.V.L.), University of Colorado, Anschutz Medical Campus, Aurora., Enyart BT; School of Medicine, Consortium for Fibrosis Research & Translation (B.T.E., K.S.M., R.A.N., K.A.K., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora.; Division of Cardiology, Department of Medicine (B.T.E., K.S.M., K.A.K.), University of Colorado, Anschutz Medical Campus, Aurora., Jolly AJ; From the Division of Renal Diseases and Hypertension, Department of Medicine (K.A.S., S.L., M.F.M., A.J.J., A.M.D., R.A.N., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora., Dubner AM; From the Division of Renal Diseases and Hypertension, Department of Medicine (K.A.S., S.L., M.F.M., A.J.J., A.M.D., R.A.N., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora., Moulton KS; School of Medicine, Consortium for Fibrosis Research & Translation (B.T.E., K.S.M., R.A.N., K.A.K., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora.; Division of Cardiology, Department of Medicine (B.T.E., K.S.M., K.A.K.), University of Colorado, Anschutz Medical Campus, Aurora., Nemenoff RA; From the Division of Renal Diseases and Hypertension, Department of Medicine (K.A.S., S.L., M.F.M., A.J.J., A.M.D., R.A.N., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora.; School of Medicine, Consortium for Fibrosis Research & Translation (B.T.E., K.S.M., R.A.N., K.A.K., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora., Koch KA; School of Medicine, Consortium for Fibrosis Research & Translation (B.T.E., K.S.M., R.A.N., K.A.K., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora.; Division of Cardiology, Department of Medicine (B.T.E., K.S.M., K.A.K.), University of Colorado, Anschutz Medical Campus, Aurora., LaBarbera DV; School of Pharmacy and Pharmaceutical Sciences (L.L., Q.Z., D.V.L.), University of Colorado, Anschutz Medical Campus, Aurora., Weiser-Evans MCM; From the Division of Renal Diseases and Hypertension, Department of Medicine (K.A.S., S.L., M.F.M., A.J.J., A.M.D., R.A.N., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora.; School of Medicine, Consortium for Fibrosis Research & Translation (B.T.E., K.S.M., R.A.N., K.A.K., M.C.M.W.-E.), University of Colorado, Anschutz Medical Campus, Aurora.
Source: Arteriosclerosis, thrombosis, and vascular biology [Arterioscler Thromb Vasc Biol] 2020 Aug; Vol. 40 (8), pp. 1854-1869. Date of Electronic Publication: 2020 Jun 25.
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Lippincott Williams & Wilkins Country of Publication: United States NLM ID: 9505803 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1524-4636 (Electronic) Linking ISSN: 10795642 NLM ISO Abbreviation: Arterioscler Thromb Vasc Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1524-4636
DOI:10.1161/ATVBAHA.120.314458