Structural Basis for α-Helix Mimicry and Inhibition of Protein-Protein Interactions with Oligourea Foldamers.

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Title: Structural Basis for α-Helix Mimicry and Inhibition of Protein-Protein Interactions with Oligourea Foldamers.
Authors: Cussol L; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France., Mauran-Ambrosino L; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France.; Ureka Pharma SAS, 2 rue Robert Escarpit, F-33607, Pessac, France., Buratto J; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France., Belorusova AY; Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), INSERM, U1258/CNRS, UMR 7104/, Univ. Strasbourg, 67404, Illkirch, France., Neuville M; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France.; Ureka Pharma SAS, 2 rue Robert Escarpit, F-33607, Pessac, France., Osz J; Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), INSERM, U1258/CNRS, UMR 7104/, Univ. Strasbourg, 67404, Illkirch, France., Fribourg S; ARNA Laboratory, INSERM U1212, UMR CNRS 5320, Univ. Bordeaux, Bordeaux, France., Fremaux J; Ureka Pharma SAS, 2 rue Robert Escarpit, F-33607, Pessac, France., Dolain C; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France., Goudreau SR; Ureka Pharma SAS, 2 rue Robert Escarpit, F-33607, Pessac, France., Rochel N; Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), INSERM, U1258/CNRS, UMR 7104/, Univ. Strasbourg, 67404, Illkirch, France., Guichard G; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France.
Source: Angewandte Chemie (International ed. in English) [Angew Chem Int Ed Engl] 2021 Feb 01; Vol. 60 (5), pp. 2296-2303. Date of Electronic Publication: 2020 Dec 01.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 0370543 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-3773 (Electronic) Linking ISSN: 14337851 NLM ISO Abbreviation: Angew Chem Int Ed Engl Subsets: MEDLINE
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  Data: Structural Basis for α-Helix Mimicry and Inhibition of Protein-Protein Interactions with Oligourea Foldamers.
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  Data: <searchLink fieldCode="AU" term="%22Cussol+L%22">Cussol L</searchLink>; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France.<br /><searchLink fieldCode="AU" term="%22Mauran-Ambrosino+L%22">Mauran-Ambrosino L</searchLink>; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France.; Ureka Pharma SAS, 2 rue Robert Escarpit, F-33607, Pessac, France.<br /><searchLink fieldCode="AU" term="%22Buratto+J%22">Buratto J</searchLink>; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France.<br /><searchLink fieldCode="AU" term="%22Belorusova+AY%22">Belorusova AY</searchLink>; Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), INSERM, U1258/CNRS, UMR 7104/, Univ. Strasbourg, 67404, Illkirch, France.<br /><searchLink fieldCode="AU" term="%22Neuville+M%22">Neuville M</searchLink>; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France.; Ureka Pharma SAS, 2 rue Robert Escarpit, F-33607, Pessac, France.<br /><searchLink fieldCode="AU" term="%22Osz+J%22">Osz J</searchLink>; Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), INSERM, U1258/CNRS, UMR 7104/, Univ. Strasbourg, 67404, Illkirch, France.<br /><searchLink fieldCode="AU" term="%22Fribourg+S%22">Fribourg S</searchLink>; ARNA Laboratory, INSERM U1212, UMR CNRS 5320, Univ. Bordeaux, Bordeaux, France.<br /><searchLink fieldCode="AU" term="%22Fremaux+J%22">Fremaux J</searchLink>; Ureka Pharma SAS, 2 rue Robert Escarpit, F-33607, Pessac, France.<br /><searchLink fieldCode="AU" term="%22Dolain+C%22">Dolain C</searchLink>; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France.<br /><searchLink fieldCode="AU" term="%22Goudreau+SR%22">Goudreau SR</searchLink>; Ureka Pharma SAS, 2 rue Robert Escarpit, F-33607, Pessac, France.<br /><searchLink fieldCode="AU" term="%22Rochel+N%22">Rochel N</searchLink>; Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), INSERM, U1258/CNRS, UMR 7104/, Univ. Strasbourg, 67404, Illkirch, France.<br /><searchLink fieldCode="AU" term="%22Guichard+G%22">Guichard G</searchLink>; Univ. Bordeaux, CNRS, Bordeaux INP, CBMN, UMR 5248, Institut Européen de Chimie et Biologie, 2 rue Robert Escarpit, F-33607, Pessac, France.
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