Snapshots and ensembles of BTK and cIAP1 protein degrader ternary complexes.

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Title: Snapshots and ensembles of BTK and cIAP1 protein degrader ternary complexes.
Authors: Schiemer J; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Horst R; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Meng Y; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Montgomery JI; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Xu Y; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Feng X; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Borzilleri K; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Uccello DP; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Leverett C; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Brown S; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Che Y; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Brown MF; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Hayward MM; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Gilbert AM; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Noe MC; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA., Calabrese MF; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, CT, USA. matthew.calabrese@pfizer.com.
Source: Nature chemical biology [Nat Chem Biol] 2021 Feb; Vol. 17 (2), pp. 152-160. Date of Electronic Publication: 2020 Nov 16.
Publication Type: Journal Article
Journal Info: Publisher: Nature Pub. Group Country of Publication: United States NLM ID: 101231976 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1552-4469 (Electronic) Linking ISSN: 15524450 NLM ISO Abbreviation: Nat Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1552-4469
DOI:10.1038/s41589-020-00686-2