Evaluation of Prediction Accuracy for Volume of Distribution in Rat and Human Using In Vitro, In Vivo, PBPK and QSAR Methods.

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Title: Evaluation of Prediction Accuracy for Volume of Distribution in Rat and Human Using In Vitro, In Vivo, PBPK and QSAR Methods.
Authors: Mathew S; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Cambridge, MA 02139, USA., Tess D; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Cambridge, MA 02139, USA., Burchett W; Early Clinical Development, Pfizer Worldwide Research and Development, Groton, CT 06340, USA., Chang G; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA., Woody N; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA., Keefer C; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA., Orozco C; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA., Lin J; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA., Jordan S; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA., Yamazaki S; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, San Diego, CA 92121, USA., Jones R; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, San Diego, CA 92121, USA., Di L; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA. Electronic address: li.di@pfizer.com.
Source: Journal of pharmaceutical sciences [J Pharm Sci] 2021 Apr; Vol. 110 (4), pp. 1799-1823. Date of Electronic Publication: 2020 Dec 16.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 2985195R Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-6017 (Electronic) Linking ISSN: 00223549 NLM ISO Abbreviation: J Pharm Sci Subsets: MEDLINE
Database: MEDLINE Ultimate
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PubType: Academic Journal
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  Data: Evaluation of Prediction Accuracy for Volume of Distribution in Rat and Human Using In Vitro, In Vivo, PBPK and QSAR Methods.
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  Data: <searchLink fieldCode="AU" term="%22Mathew+S%22">Mathew S</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Cambridge, MA 02139, USA.<br /><searchLink fieldCode="AU" term="%22Tess+D%22">Tess D</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Cambridge, MA 02139, USA.<br /><searchLink fieldCode="AU" term="%22Burchett+W%22">Burchett W</searchLink>; Early Clinical Development, Pfizer Worldwide Research and Development, Groton, CT 06340, USA.<br /><searchLink fieldCode="AU" term="%22Chang+G%22">Chang G</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA.<br /><searchLink fieldCode="AU" term="%22Woody+N%22">Woody N</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA.<br /><searchLink fieldCode="AU" term="%22Keefer+C%22">Keefer C</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA.<br /><searchLink fieldCode="AU" term="%22Orozco+C%22">Orozco C</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA.<br /><searchLink fieldCode="AU" term="%22Lin+J%22">Lin J</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA.<br /><searchLink fieldCode="AU" term="%22Jordan+S%22">Jordan S</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA.<br /><searchLink fieldCode="AU" term="%22Yamazaki+S%22">Yamazaki S</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, San Diego, CA 92121, USA.<br /><searchLink fieldCode="AU" term="%22Jones+R%22">Jones R</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, San Diego, CA 92121, USA.<br /><searchLink fieldCode="AU" term="%22Di+L%22">Di L</searchLink>; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, CT 06340, USA. Electronic address: li.di@pfizer.com.
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  Data: <searchLink fieldCode="JN" term="%222985195R%22">Journal of pharmaceutical sciences</searchLink> [J Pharm Sci] 2021 Apr; Vol. 110 (4), pp. 1799-1823. <i>Date of Electronic Publication: </i>2020 Dec 16.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier%22">Elsevier </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>2985195R <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-6017 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200223549%22">00223549 </searchLink><i>NLM ISO Abbreviation: </i>J Pharm Sci <i>Subsets: </i>MEDLINE
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        Value: 10.1016/j.xphs.2020.12.005
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              Text: 2021 Apr
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