Parallel discovery of selective and dual inhibitors of tryptophan dioxygenases IDO1 and TDO2 with a newly-modified enzymatic assay.

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Title: Parallel discovery of selective and dual inhibitors of tryptophan dioxygenases IDO1 and TDO2 with a newly-modified enzymatic assay.
Authors: Capochiani de Iudicibus R; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: r.capochiani@auckland.ac.nz., Tomek P; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: p.tomek@auckland.ac.nz., Palmer BD; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: b.palmer@auckland.ac.nz., Tijono SM; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: s.tijono@auckland.ac.nz., Flanagan JU; Department of Pharmacology and Clinical Pharmacology, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: j.flanagan@auckland.ac.nz., Ching LM; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: l.ching@auckland.ac.nz.
Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2021 Jun 01; Vol. 39, pp. 116160. Date of Electronic Publication: 2021 Apr 20.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3391 (Electronic) Linking ISSN: 09680896 NLM ISO Abbreviation: Bioorg Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: <searchLink fieldCode="AU" term="%22Capochiani+de+Iudicibus+R%22">Capochiani de Iudicibus R</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: r.capochiani@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Tomek+P%22">Tomek P</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: p.tomek@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Palmer+BD%22">Palmer BD</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: b.palmer@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Tijono+SM%22">Tijono SM</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: s.tijono@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Flanagan+JU%22">Flanagan JU</searchLink>; Department of Pharmacology and Clinical Pharmacology, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: j.flanagan@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Ching+LM%22">Ching LM</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: l.ching@auckland.ac.nz.
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              Text: 2021 Jun 01
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