Parallel discovery of selective and dual inhibitors of tryptophan dioxygenases IDO1 and TDO2 with a newly-modified enzymatic assay.
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| Title: | Parallel discovery of selective and dual inhibitors of tryptophan dioxygenases IDO1 and TDO2 with a newly-modified enzymatic assay. |
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| Authors: | Capochiani de Iudicibus R; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: r.capochiani@auckland.ac.nz., Tomek P; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: p.tomek@auckland.ac.nz., Palmer BD; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: b.palmer@auckland.ac.nz., Tijono SM; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: s.tijono@auckland.ac.nz., Flanagan JU; Department of Pharmacology and Clinical Pharmacology, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: j.flanagan@auckland.ac.nz., Ching LM; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: l.ching@auckland.ac.nz. |
| Source: | Bioorganic & medicinal chemistry [Bioorg Med Chem] 2021 Jun 01; Vol. 39, pp. 116160. Date of Electronic Publication: 2021 Apr 20. |
| Publication Type: | Journal Article; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3391 (Electronic) Linking ISSN: 09680896 NLM ISO Abbreviation: Bioorg Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 33901770 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Parallel discovery of selective and dual inhibitors of tryptophan dioxygenases IDO1 and TDO2 with a newly-modified enzymatic assay. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Capochiani+de+Iudicibus+R%22">Capochiani de Iudicibus R</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: r.capochiani@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Tomek+P%22">Tomek P</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: p.tomek@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Palmer+BD%22">Palmer BD</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: b.palmer@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Tijono+SM%22">Tijono SM</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: s.tijono@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Flanagan+JU%22">Flanagan JU</searchLink>; Department of Pharmacology and Clinical Pharmacology, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: j.flanagan@auckland.ac.nz.<br /><searchLink fieldCode="AU" term="%22Ching+LM%22">Ching LM</searchLink>; Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, University of Auckland, The University of Auckland, Private Bag 92019, Victoria Street West, Auckland 1142, New Zealand. Electronic address: l.ching@auckland.ac.nz. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229413298%22">Bioorganic & medicinal chemistry</searchLink> [Bioorg Med Chem] 2021 Jun 01; Vol. 39, pp. 116160. <i>Date of Electronic Publication: </i>2021 Apr 20. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Research Support, Non-U.S. Gov't – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science%22">Elsevier Science </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9413298 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3391 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2209680896%22">09680896 </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=33901770 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmc.2021.116160 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 116160 Titles: – TitleFull: Parallel discovery of selective and dual inhibitors of tryptophan dioxygenases IDO1 and TDO2 with a newly-modified enzymatic assay. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Capochiani de Iudicibus R – PersonEntity: Name: NameFull: Tomek P – PersonEntity: Name: NameFull: Palmer BD – PersonEntity: Name: NameFull: Tijono SM – PersonEntity: Name: NameFull: Flanagan JU – PersonEntity: Name: NameFull: Ching LM IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 06 Text: 2021 Jun 01 Type: published Y: 2021 Identifiers: – Type: issn-electronic Value: 1464-3391 Numbering: – Type: volume Value: 39 Titles: – TitleFull: Bioorganic & medicinal chemistry Type: main |
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