Rapid Evaluation of Small Molecule Cellular Target Engagement with a Luminescent Thermal Shift Assay.

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Bibliographic Details
Title: Rapid Evaluation of Small Molecule Cellular Target Engagement with a Luminescent Thermal Shift Assay.
Authors: Mortison JD; Chemical Biology, Merck & Co., Inc., Boston, Massachusetts 02115, United States., Cornella-Taracido I; Chemical Biology, Merck & Co., Inc., Boston, Massachusetts 02115, United States., Venkatchalam G; Quantitative Biosciences, MSD, Singapore 138665, Singapore., Partridge AW; Quantitative Biosciences, MSD, Singapore 138665, Singapore., Siriwardana N; Chemical Biology, Merck & Co., Inc., Boston, Massachusetts 02115, United States., Bushell SM; Chemical Biology, Merck & Co., Inc., Boston, Massachusetts 02115, United States.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2021 Jul 12; Vol. 12 (8), pp. 1288-1294. Date of Electronic Publication: 2021 Jul 12 (Print Publication: 2021).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1948-5875
DOI:10.1021/acsmedchemlett.1c00276