Suppression of Colon Tumorigenesis in Mutant Apc Mice by a Novel PDE10 Inhibitor that Reduces Oncogenic β-Catenin.

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Title: Suppression of Colon Tumorigenesis in Mutant Apc Mice by a Novel PDE10 Inhibitor that Reduces Oncogenic β-Catenin.
Authors: Lee KJ; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Chang WL; Cancer Prevention and Control Program, Fox Chase Cancer Center, Philadelphia, Pennsylvania., Chen X; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Valiyaveettil J; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Ramirez-Alcantara V; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Gavin E; Gynecologic Oncology Research Division, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Musiyenko A; Gynecologic Oncology Research Division, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Madeira da Silva L; Gynecologic Oncology Research Division, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Annamdevula NS; Department of Chemical and Biomedical Engineering, University of South Alabama, Mobile, Alabama.; Center for Lung Biology, University of South Alabama, Mobile, Alabama., Leavesley SJ; Department of Chemical and Biomedical Engineering, University of South Alabama, Mobile, Alabama.; Center for Lung Biology, University of South Alabama, Mobile, Alabama.; Department of Pharmacology, University of South Alabama, Mobile, Alabama., Ward A; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Mattox T; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Lindsey AS; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Andrews J; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Zhu B; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Wood C; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Neese A; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Nguyen A; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Berry K; Drug Discovery Research Center, Mitchell Cancer Institute, University of South Alabama, Mobile, Alabama., Maxuitenko Y; Department of Drug Discovery and Development, Harrison School of Pharmacy, Auburn University, Auburn, Alabama., Moyer MP; INCELL Corporation LLC, San Antonio, Texas., Nurmemmedov E; Saint John's Cancer Institute, Santa Monica, California., Gorman G; Samford University, Birmingham, Alabama., Coward L; Samford University, Birmingham, Alabama., Zhou G; Georgia Cancer Center, Augusta University, Augusta, Georgia., Keeton AB; Department of Drug Discovery and Development, Harrison School of Pharmacy, Auburn University, Auburn, Alabama., Cooper HS; Department of Pathology, Fox Chase Cancer Center, Philadelphia, Pennsylvania., Clapper ML; Cancer Prevention and Control Program, Fox Chase Cancer Center, Philadelphia, Pennsylvania., Piazza GA; Department of Drug Discovery and Development, Harrison School of Pharmacy, Auburn University, Auburn, Alabama. gap0034@auburn.edu.
Source: Cancer prevention research (Philadelphia, Pa.) [Cancer Prev Res (Phila)] 2021 Nov; Vol. 14 (11), pp. 995-1008. Date of Electronic Publication: 2021 Sep 28.
Publication Type: Journal Article; Research Support, N.I.H., Extramural
Journal Info: Publisher: American Association for Cancer Research Country of Publication: United States NLM ID: 101479409 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1940-6215 (Electronic) Linking ISSN: 19406215 NLM ISO Abbreviation: Cancer Prev Res (Phila) Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1940-6215
DOI:10.1158/1940-6207.CAPR-21-0208